Inhibition of the HERG channel by droperidol depends on channel gating and involves the S6 residue F656

Anesthesia and Analgesia

Volumn 106, Issue 4, 2008, Pages 1161-1170

  Luo, Tao ^a,b   Luo, Ailin ^b   Liu, Miu ^a   Liu, Xianyi ^a  

^a RENMIN HOSPITAL OF WUHAN UNIVERSITY   (China)

^b HUAZHONG UNIVERSITY OF SCIENCE AND TECHNOLOGY   (China)

Author keywords

[No Author keywords available]

Indexed keywords

DROPERIDOL; METHIONINE; PHENYLALANINE; POTASSIUM CHANNEL HERG; PROTEIN S6; SERINE; THREONINE;

ARTICLE; CELL MEMBRANE POTENTIAL; CELL STRAIN HEK293; CHANNEL GATING; CONTROLLED STUDY; GENE MUTATION; HUMAN; HUMAN CELL; INHIBITION KINETICS; PATCH CLAMP; PRIORITY JOURNAL; PROTEIN BINDING; PROTEIN EXPRESSION; STEADY STATE; WHOLE CELL;

CELL LINE; DROPERIDOL; ELECTROPHYSIOLOGY; ETHER-A-GO-GO POTASSIUM CHANNELS; HUMANS; ION CHANNEL GATING; KIDNEY; KINETICS; PATCH-CLAMP TECHNIQUES; TRANSFECTION;

EID: 41349122946     PISSN: 00032999     EISSN: None     Source Type: Journal    
DOI: 10.1213/ane.0b013e3181684974     Document Type: Article

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