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Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 5, 2008, Pages 1617-1622

4,4-Dimethyl-1,2,3,4-tetrahydroquinoline-based PPARα/γ agonists. Part I: Synthesis and pharmacological evaluation

(10) Parmenon, Cécile a Guillard, Jérôme a Caignard, Daniel Henri b Hennuyer, Nathalie c Staels, Bart c Audinot Bouchez, Valérie d Boutin, Jean Albert d Dacquet, Catherine e Ktorza, Alain e Viaud Massuard, Marie Claude a

a UFR des Sciences Pharmaceutiques (France)

b INSTITUT DE RECHERCHES SERVIER (France)

c INSTITUT PASTEUR DE LILLE (France)

d Division de Recherche Pharmacologie Moléculaire et Cellulaire (France)

e INSTITUT DE RECHERCHES SERVIER (France)

Author keywords

4,4 Dimethyl 1,2,3,4 tetrahydroquinoline; Diabetes type 2; PPAR agonists

Indexed keywords

4,4 DIMETHYL 1,2,3,4 TETRAHYDROQUINOLINE; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR AGONIST; PEROXISOME PROLIFERATOR ACTIVATED RECEPTOR GAMMA; ROSIGLITAZONE; TESAGLITAZAR; UNCLASSIFIED DRUG;

ARTICLE; DRUG ACTIVITY; DRUG BINDING; DRUG SYNTHESIS;

EID: 39849086207 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/j.bmcl.2008.01.067 Document Type: Article

Times cited : (40)

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