Anti-Pneumocystis carinii and antiplasmodial activities of primaquine-derived imidazolidin-4-ones

Bioorganic and Medicinal Chemistry Letters

Volumn 18, Issue 2, 2008, Pages 485-488

  Vale, Nuno ^a   Collins, Margaret S ^c,d   Gut, Jiri ^e   Ferraz, Ricardo ^a,b   Rosenthal, Philip J ^e   Cushion, Melanie T ^c,d   Moreira, Rui ^f   Gomes, Paula ^a  

^a UNIVERSITY OF PORTO   (Portugal)

^b POLYTECHNIC INSTITUTE OF PORTO   (Portugal)

^c UNIVERSITY OF CINCINNATI COLLEGE OF MEDICINE   (United States)

^d VETERANS AFFAIRS MEDICAL CENTER   (United States)

^e UNIVERSITY OF CALIFORNIA   (United States)

^f RESEARCH INSTITUTE FOR MEDICINES IMED ULISBOA   (Portugal)

Author keywords

AIDS; Antimalarial; Antiplasmodial; HIV; Infection; Malaria; Plasmodium falciparum; Pneumocystis carinii; Primaquine

Indexed keywords

8 AMINOQUINOLINE DERIVATIVE; ANTIFUNGAL AGENT; ANTIMALARIAL AGENT; IMIDAZOLIDIN 4 ONE DERIVATIVE; IMIDAZOLIDINE DERIVATIVE; PRIMAQUINE DERIVATIVE; UNCLASSIFIED DRUG;

ANIMAL CELL; ANIMAL EXPERIMENT; ANIMAL MODEL; ANIMAL TISSUE; ANTIMICROBIAL ACTIVITY; ARTICLE; CONTROLLED STUDY; DRUG ACTIVITY; DRUG SCREENING; DRUG STABILITY; IN VITRO STUDY; METABOLIC REGULATION; MOUSE; NONHUMAN; PLASMODIUM; PLASMODIUM FALCIPARUM; PLASMODIUM FALCIPARUM W2; PNEUMOCYSTIS CARINII; STRAIN IDENTIFICATION;

ANIMALS; ANTIFUNGAL AGENTS; ANTIMALARIALS; IMIDAZOLINES; MICE; MICROBIAL SENSITIVITY TESTS; PLASMODIUM FALCIPARUM; PNEUMOCYSTIS CARINII; PRIMAQUINE;

PLASMODIUM FALCIPARUM; PNEUMOCYSTIS CARINII;

EID: 38149054056     PISSN: 0960894X     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmcl.2007.11.105     Document Type: Article

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