LRET-based HTS of a small-compound library for inhibitors of bacterial RNA polymerase

Assay and Drug Development Technologies

Volumn 5, Issue 6, 2007, Pages 759-768

  Glaser, Bryan T ^a   Bergendahl, Veit ^a,b   Thompson, Nancy E ^a   Olson, Brian ^a,c   Burgess, Richard R ^a  

^a UNIVERSITY OF WISCONSIN MADISON   (United States)

^b UNIVERSITY OF WISCONSIN MADISON   (United States)

^c UNIVERSITY OF WISCONSIN   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BACTERIAL ENZYME; ENZYME INHIBITOR; RNA POLYMERASE;

ARTICLE; BACTERIAL GROWTH; DRUG DETERMINATION; ESCHERICHIA COLI; HIGH THROUGHPUT SCREENING; LUMINESCENCE; LUMINESCENCE RESONANCE ENERGY TRANSFER; NONHUMAN; RNA TRANSCRIPTION;

ANTI-BACTERIAL AGENTS; BACTERIA; DNA-DIRECTED RNA POLYMERASES; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; ESCHERICHIA COLI; FLUORESCENCE RESONANCE ENERGY TRANSFER; GENE EXPRESSION REGULATION, BACTERIAL; HELA CELLS; HUMANS; MICROBIAL SENSITIVITY TESTS;

EID: 38049071617     PISSN: 1540658X     EISSN: None     Source Type: Journal    
DOI: 10.1089/adt.2007.095     Document Type: Article

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