Development of a specific inhibitor for the placental protease, cathepsin P

Archives of Biochemistry and Biophysics

Volumn 464, Issue 2, 2007, Pages 288-294

  Hassanein, Mohamed ^a,b   Xue, Fengtian ^c   Seto, Christopher T ^c   Mason, Robert W ^a  

^a NEMOURS ALFRED I DUPONT HOSPITAL FOR CHILDREN   (United States)

^b UNIVERSITY OF DELAWARE   (United States)

^c BROWN UNIVERSITY   (United States)

Author keywords

Cathepsin; Inhibition; Kinetics; Placenta; Specificity

Indexed keywords

AROMATIC AMINO ACID; CARBOBENZYLOXYTRYPTOPHYLTRYPTOPHAN 4 CYCLOHEXANONE TRYPTOPHYLPHENYLALANINE METHYL ESTER; CATHEPSIN; CATHEPSIN B; CATHEPSIN L; CATHEPSIN P; CYCLOHEXANONE; CYCLOHEXANONE DERIVATIVE; CYSTEINE PROTEINASE; DIPEPTIDE; LYSOSOME ENZYME; POLYPEPTIDE; PROTEINASE INHIBITOR; TRYPTOPHAN; TYROSINE; UNCLASSIFIED DRUG;

ARTICLE; BIOLOGICAL ACTIVITY; COMBINATORIAL LIBRARY; ENZYME ACTIVITY; ENZYME ANALYSIS; ENZYME LOCALIZATION; ENZYME SPECIFICITY; ENZYME SUBSTRATE; HUMAN; NONHUMAN; PHARMACOPHORE; PLACENTA; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FAMILY; PROTEINASE INHIBITION;

ANIMALS; CATHEPSINS; DRUG DESIGN; FEMALE; MICE; PLACENTA; PROTEASE INHIBITORS;

RODENTIA;

EID: 34547666652     PISSN: 00039861     EISSN: 10960384     Source Type: Journal    
DOI: 10.1016/j.abb.2007.04.019     Document Type: Article

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