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Volumn 63, Issue 33, 2007, Pages 7949-7969

Synthesis of chiral β2,2,3-3-amino-2-hydroxyalkanoates and 3-alkyl-3-hydroxy-β-lactams by double asymmetric induction

Author keywords

Hydroxy amino acids; 3 Hydroxy lactams; Aldimines; Dioxolan 4 ones; Double asymmetric induction

Indexed keywords

1' AMINODIOXOLANONE DERIVATIVE; ALKANOIC ACID; ATROLACTIC ACID; BETA LACTAM DERIVATIVE; FUNCTIONAL GROUP; IMINE; LACTIC ACID DERIVATIVE; MANDELIC ACID DERIVATIVE; METHYL BETA SULFINYLAMINOPROPIONATE DERIVATIVE; N SULFINYL 1' AMINODIOXALONONE DERIVATIVE; UNCLASSIFIED DRUG;

EID: 34347211695     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.tet.2007.05.069     Document Type: Article
Times cited : (17)

References (81)
  • 6
    • 34347216437 scopus 로고    scopus 로고
    • BaMaung, N. Y.; Niles, I. L.; Craig, R. A.; Henkin, J.; Kawai, M.; Searle, X. B.; Sheppard, G. S.; Wang, J. Int. Pub. N. WO 2004/013085 A1, 12.02.2004.
  • 15
    • 34347216089 scopus 로고    scopus 로고
    • See, for example:
  • 22
    • 34347219176 scopus 로고    scopus 로고
    • For selected examples of biologically active constrained norstatines, which bear an aromatic substituent at the C3 carbon atom and a methyl at the C2, see:
  • 23
    • 37049077584 scopus 로고    scopus 로고
    • Denis, J.-N.; Fkyerat, A.; Gimbert, Y.; Coutterez, C.; Mantellier, P.; Jost, S.; Greene, A. E. J. Chem. Soc., Perkin Trans. 1 1995, 1811-1816.
  • 29
    • 34347257528 scopus 로고    scopus 로고
    • For the synthesis of BOC aldimines, see for example:
  • 36
    • 34347221290 scopus 로고    scopus 로고
    • note
    • An inversion for the descriptor of the 1′-position of 1′-aminodioxolanones which bear the heteroaromatic 2-thienyl substituent occurs, with respect to other dioxolanones, due to the priority rule at this stereocenter.
  • 38
    • 34347257882 scopus 로고    scopus 로고
    • Holton, R. A.; Nadizadeh, H.; Beidiger, R. J. Fury1 and Thienyl Substituted Taxanes as Antitumor Agents. EP 0534708A1, 1993;
  • 39
    • 34347268193 scopus 로고    scopus 로고
    • Holton, R. A.; Chai, K.-B. Idmoumaz, H.; Nadizadeh, H.; Rengan, K.; Suzuki, Y.; Tao, C. U.S. Patent 6,794,523, September 21, 2004.
  • 61
    • 34347232433 scopus 로고    scopus 로고
    • See Ref. 4a.
  • 73
  • 74
    • 34347211114 scopus 로고    scopus 로고
    • For the synthesis of N-(S)-tert-butylsulfinyl adimines, see:
  • 78
    • 0037223313 scopus 로고    scopus 로고
    • For the preparation of α-sulfonyl carbamates, see:
    • Ellman J.A. Pure Appl. Chem. 75 (2003) 39-46 For the preparation of α-sulfonyl carbamates, see:
    • (2003) Pure Appl. Chem. , vol.75 , pp. 39-46
    • Ellman, J.A.1


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.