-
1
-
-
0022448676
-
Cellular effects of cannabinoids
-
Martin BR. Cellular effects of cannabinoids. Pharmacol Rev. 1986;38:45-74.
-
(1986)
Pharmacol Rev.
, vol.38
, pp. 45-74
-
-
Martin, B.R.1
-
2
-
-
0024263922
-
Determination and characterization of a cannabinoid receptor in rat brain
-
Devane WA, Dysarz FA 3d, Johnson MR, Melvin LS, Howlett AC. Determination and characterization of a cannabinoid receptor in rat brain. Mol Pharmacol. 1988; 34:605-613.
-
(1988)
Mol Pharmacol.
, vol.34
, pp. 605-613
-
-
Devane, W.A.1
Dysarz III, F.A.2
Johnson, M.R.3
Melvin, L.S.4
Howlett, A.C.5
-
3
-
-
0027515373
-
Molecular characterization of a peripheral receptor for cannabinoids
-
Munro S, Thomas KL, Abu-Shaar M. Molecular characterization of a peripheral receptor for cannabinoids. Nature (London) 1993;365:61-65.
-
(1993)
Nature (London)
, vol.365
, pp. 61-65
-
-
Munro, S.1
Thomas, K.L.2
Abu-Shaar, M.3
-
4
-
-
0344058079
-
-
US Patent 5,624,941 Apr. 29
-
Barth F, Casellas P, Congy C, Martinez S, Rinaldi M, Anne-Archard G. Pyrazole derivatives, method of preparing them and pharmaceutical compositions in which they are present. US Patent 5,624,941 Apr. 29, 1997.
-
(1997)
Pyrazole Derivatives, Method of Preparing Them and Pharmaceutical Compositions in Which They Are Present
-
-
Barth, F.1
Casellas, P.2
Congy, C.3
Martinez, S.4
Rinaldi, M.5
Anne-Archard, G.6
-
5
-
-
0028129936
-
SR141716A, a potent and selective antagonist of the brain cannabinoid receptor
-
Rinaldi-Carmona M, Barth F, Héaulme M, Shire D, Calandra B, Congy C, Martinez S, Maruani J, Néliat G, Caput D, Ferrara P, Soubrié P, Breliere JC, Le Fur G. SR141716A, A potent and selective antagonist of the brain cannabinoid receptor. FEBS Lett. 1994;350:240-244.
-
(1994)
FEBS Lett.
, vol.350
, pp. 240-244
-
-
Rinaldi-Carmona, M.1
Barth, F.2
Héaulme, M.3
Shire, D.4
Calandra, B.5
Congy, C.6
Martinez, S.7
Maruani, J.8
Néliat, G.9
Caput, D.10
Ferrara, P.11
Soubrié, P.12
Breliere, J.C.13
Le Fur, G.14
-
6
-
-
0029034879
-
Biochemical and pharmacological characterization of SR141716A, the first potent and selective brain cannabinoid receptor antagonist
-
Rinaldi-Carmona M, Barth F, Héaulme M, Alonso R, Shire D, Congy C, Soubrié P, Breliere JC, Le Fur G. Biochemical and pharmacological characterization of SR141716A, the first potent and selective brain cannabinoid receptor antagonist. Life Sci. 1995;56:1941-1947.
-
(1995)
Life Sci.
, vol.56
, pp. 1941-1947
-
-
Rinaldi-Carmona, M.1
Barth, F.2
Héaulme, M.3
Alonso, R.4
Shire, D.5
Congy, C.6
Soubrié, P.7
Breliere, J.C.8
Le Fur, G.9
-
7
-
-
0029965292
-
Structural features of the central cannabinoid CB1 receptor involved in the binding of the specific CB1 antagonist SR 141716A
-
Shire D, Calandra B, Delpech M, Dumont X, Kaghad M, Le Fur G, Caput D, Ferrara P. Structural features of the central cannabinoid CB1 receptor involved in the binding of the specific CB1 antagonist SR 141716A. J Biol Chem. 1996;271:6941-6946.
-
(1996)
J Biol Chem.
, vol.271
, pp. 6941-6946
-
-
Shire, D.1
Calandra, B.2
Delpech, M.3
Dumont, X.4
Kaghad, M.5
Le Fur, G.6
Caput, D.7
Ferrara, P.8
-
8
-
-
0029912522
-
Characterization and distribution of binding sites for [3H]-SR 141716A, a selective brain (CB1) cannabinoid receptor antagonist, in rodent brain
-
Rinaldi-Carmona M, Pialot F, Congy C, Redon E, Barth F, Bachy A, Breliere JC, Soubrié P, Le Fur G. Characterization and distribution of binding sites for [3H]-SR 141716A, a selective brain (CB1) cannabinoid receptor antagonist, in rodent brain. Life Sci. 1996;58:1239-1247.
-
(1996)
Life Sci.
, vol.58
, pp. 1239-1247
-
-
Rinaldi-Carmona, M.1
Pialot, F.2
Congy, C.3
Redon, E.4
Barth, F.5
Bachy, A.6
Breliere, J.C.7
Soubrié, P.8
Le Fur, G.9
-
10
-
-
0029798021
-
Preparation of iodine-123 labeled AM251: A potential SPECT radioligand for the brain cannabinoid CB1 receptor
-
Lan R, Galley SJ, Makriyannis A. Preparation of iodine-123 labeled AM251: a potential SPECT radioligand for the brain cannabinoid CB1 receptor. J Label Compds Radiopharma 1996;38:875-881.
-
(1996)
J Label Compds Radiopharma
, vol.38
, pp. 875-881
-
-
Lan, R.1
Galley, S.J.2
Makriyannis, A.3
-
11
-
-
4143108422
-
Binding of the non-classical cannabinoid CP 55,940, and the diarylpyrazole AM251 to rodent brain cannabinoid receptors
-
Galley SJ, Lan R, Pyatt B, Gifford AN, Volkow ND, Makriyannis A. Binding of the non-classical cannabinoid CP 55,940, and the diarylpyrazole AM251 to rodent brain cannabinoid receptors. Life Sci. 1997;61:PL191-197.
-
(1997)
Life Sci.
, vol.61
-
-
Galley, S.J.1
Lan, R.2
Pyatt, B.3
Gifford, A.N.4
Volkow, N.D.5
Makriyannis, A.6
-
12
-
-
0025236913
-
Cannabinoid receptor localization in brain
-
Herkenham M, Lynn AB, Little MD, Johnson MR, Melvin LS, DeCosla BR, Rice KC. Cannabinoid receptor localization in brain. Proc Nail Acad Sci. 1990;87:1932-1936.
-
(1990)
Proc Nail Acad Sci.
, vol.87
, pp. 1932-1936
-
-
Herkenham, M.1
Lynn, A.B.2
Little, M.D.3
Johnson, M.R.4
Melvin, L.S.5
DeCosla, B.R.6
Rice, K.C.7
-
13
-
-
0025954862
-
Characterization and localization of cannabinoid receptors in rat brain: A quantitative in vitro auloradiographic study
-
Herkenham M, Lynn AB, Johnson MR, Melvin LS, DeCosta BR, Rice KC. Characterization and localization of cannabinoid receptors in rat brain: a quantitative in vitro auloradiographic study. J Neurosci. 1991;11:563-583.
-
(1991)
J Neurosci.
, vol.11
, pp. 563-583
-
-
Herkenham, M.1
Lynn, A.B.2
Johnson, M.R.3
Melvin, L.S.4
DeCosta, B.R.5
Rice, K.C.6
-
14
-
-
0031972639
-
Imaging the brain marijuana receptor: Development of a radioligand that binds to cannabinoid CB1 receptors in vivo
-
Galley SJ, Lan R, Volkow ND, Pappas N, King P, Wong CT, Gifford AN, Pyatt B, Dewey SL, Makriyannis A. Imaging the brain marijuana receptor: Development of a radioligand that binds to cannabinoid CB1 receptors in vivo. J Neurochem. 1998; 70:417-23.
-
(1998)
J Neurochem.
, vol.70
, pp. 417-423
-
-
Galley, S.J.1
Lan, R.2
Volkow, N.D.3
Pappas, N.4
King, P.5
Wong, C.T.6
Gifford, A.N.7
Pyatt, B.8
Dewey, S.L.9
Makriyannis, A.10
-
15
-
-
0023185831
-
Eleclrophilic destannylation: Stereospecific introduction of electrophiles at the 21 position of (17α)-19-Norpregna-1,3,5(10),20-tetraene-3-17β-diols
-
Hanson RN, El-Wakil H. Eleclrophilic destannylation: stereospecific introduction of electrophiles at the 21 position of (17α)-19-Norpregna-1,3,5(10),20-tetraene-3-17β-diols. J Org Chem. 1987;52:3687-3688.
-
(1987)
J Org Chem.
, vol.52
, pp. 3687-3688
-
-
Hanson, R.N.1
El-Wakil, H.2
-
16
-
-
0029786781
-
Further evidence for the presence of cannabinoid CB1 receptors in guinea-pig small intestine
-
Pertwee, RG, Fernando, SR, Nash, JE, Coutts, AA. Further evidence for the presence of cannabinoid CB1 receptors in guinea-pig small intestine. Br J Pharmacol. 1996;118:2199-2205.
-
(1996)
Br J Pharmacol.
, vol.118
, pp. 2199-2205
-
-
Pertwee, R.G.1
Fernando, S.R.2
Nash, J.E.3
Coutts, A.A.4
-
17
-
-
0031473751
-
Effect of the cannabinoid receptor SPECT agent, AM 281, on hippocampal acelylcholine release from rat brain slices
-
Gifford AN, Tang Y, Galley SJ, Volkow ND, Lan R, Makriyannis A. Effect of the cannabinoid receptor SPECT agent, AM 281, on hippocampal acelylcholine release from rat brain slices. Neurosci Lett. 1997;238:84-86.
-
(1997)
Neurosci Lett.
, vol.238
, pp. 84-86
-
-
Gifford, A.N.1
Tang, Y.2
Galley, S.J.3
Volkow, N.D.4
Lan, R.5
Makriyannis, A.6
-
18
-
-
0032505136
-
Classical/nonclassical hydrid cannabinoids: Southern aliphatic chain-funclionalized C-6β methyl, ethyl, and propyl analogues
-
Drake DJ, Jensen RS, Busch-Peterson J, Kawakami JK, Fernandez-Garcia MC, Fan P, Makriyannis A, Tius MA. Classical/nonclassical hydrid cannabinoids: southern aliphatic chain-funclionalized C-6β methyl, ethyl, and propyl analogues. J Med Chem. 1998;41:3596-3608.
-
(1998)
J Med Chem.
, vol.41
, pp. 3596-3608
-
-
Drake, D.J.1
Jensen, R.S.2
Busch-Peterson, J.3
Kawakami, J.K.4
Fernandez-Garcia, M.C.5
Fan, P.6
Makriyannis, A.7
Tius, M.A.8
-
19
-
-
0028246688
-
(R)-methanandamide: A chiral novel anandamide possessing higher potency and metabolic stability
-
Abadji V, Lin S, Taha G, Griffin G, Stevenson LA, Pertwee RG, Makriyannis A. (R)-methanandamide: a chiral novel anandamide possessing higher potency and metabolic stability. J Med Chem. 1994;37:1889-1893.
-
(1994)
J Med Chem.
, vol.37
, pp. 1889-1893
-
-
Abadji, V.1
Lin, S.2
Taha, G.3
Griffin, G.4
Stevenson, L.A.5
Pertwee, R.G.6
Makriyannis, A.7
-
20
-
-
0019791636
-
A rapid method for preparing synaptosomes: Comparison, with alternative procedures
-
Dodd PR, Hardy JA, Oakley AE, Edwardson JA, Perry EK, Delaunoy JP. A rapid method for preparing synaptosomes: comparison, with alternative procedures. Brain Res. 1981;226:107-118.
-
(1981)
Brain Res.
, vol.226
, pp. 107-118
-
-
Dodd, P.R.1
Hardy, J.A.2
Oakley, A.E.3
Edwardson, J.A.4
Perry, E.K.5
Delaunoy, J.P.6
-
22
-
-
0015861774
-
Relationship between the inhibition constant (Ki) and the concentration of inhibitor which causes 50 per cent (IC50) of an enzymatic reaction
-
50) of an enzymatic reaction. Biochem Pharmacol. 1973;22:3099-3108.
-
(1973)
Biochem Pharmacol.
, vol.22
, pp. 3099-3108
-
-
Cheng, Y.1
Prusoff, W.H.2
-
23
-
-
0030814261
-
Inhibition by cannabinoid receptor agonists of acetylcholine release from the guinea-pig Myenteric plexus
-
Coutts AA, Pertwee RG. Inhibition by cannabinoid receptor agonists of acetylcholine release from the guinea-pig Myenteric plexus. Br J Pharmacol. 1997;21:1557-1566.
-
(1997)
Br J Pharmacol.
, vol.21
, pp. 1557-1566
-
-
Coutts, A.A.1
Pertwee, R.G.2
-
24
-
-
0018655874
-
pA2 and receptor differentiation: A statistical analysis of competitive antagonism
-
Tallarida RJ, Cowan A, Adler MW. pA2 and receptor differentiation: a statistical analysis of competitive antagonism. Life Sci. 1979;25:637-654.
-
(1979)
Life Sci.
, vol.25
, pp. 637-654
-
-
Tallarida, R.J.1
Cowan, A.2
Adler, M.W.3
|