123I-labeled AM251: A radioiodinated ligand which binds in vivo to mouse brain cannabinoid CB1 receptors

European Journal of Pharmacology

Volumn 307, Issue 3, 1996, Pages 331-338

  Gatley, S John ^a   Gifford, Andrew N ^a   Volkow, Nora D ^a   Lan, Ruoxi ^b   Makriyannis, Alexandros ^b  

^a BROOKHAVEN NATIONAL LABORATORY   (United States)

^b UNIVERSITY OF CONNECTICUT   (United States)

Author keywords

Canabinoid receptor antagonist; SR141617A; 9 Tetrahydrocannabinol

Indexed keywords

1 (2,4 DICHLOROPHENYL) 5 (4 IODOPHENYL) 4 METHYL N (1 PIPERIDYL) 1H PYRAZOLE 3 CARBOXAMIDE; BRAIN RECEPTOR; CANNABINOID RECEPTOR; IODINE 123; PIPERIDINE DERIVATIVE; PYRAZOLE DERIVATIVE; RECEPTOR SUBTYPE; RIMONABANT; UNCLASSIFIED DRUG; DIAGNOSTIC AGENT; DRUG RECEPTOR; RADIOACTIVE IODINE; TETRAHYDROCANNABINOL;

ANIMAL EXPERIMENT; ANIMAL TISSUE; ARTICLE; BRAIN; CONTROLLED STUDY; DRUG RECEPTOR BINDING; INTRAVENOUS DRUG ADMINISTRATION; ISOTOPE LABELING; LIGAND BINDING; MALE; MOUSE; NONHUMAN; PRIORITY JOURNAL; RADIOIODINATION; TISSUE DISTRIBUTION; ANIMAL; BLOOD; CELL MEMBRANE; DRUG ANTAGONISM; DRUG EFFECT; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; HIPPOCAMPUS; METABOLISM; MOTOR ACTIVITY; MOUSE STRAIN; PROTEIN BINDING; RADIOASSAY; ULTRASTRUCTURE;

ANIMALS; BRAIN; CELL MEMBRANE; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; HIPPOCAMPUS; IODINE RADIOISOTOPES; ISOTOPE LABELING; MALE; MICE; MICE, INBRED STRAINS; MOTOR ACTIVITY; PIPERIDINES; PROTEIN BINDING; PYRAZOLES; RADIOLIGAND ASSAY; RECEPTORS, CANNABINOID; RECEPTORS, DRUG; TETRAHYDROCANNABINOL; TISSUE DISTRIBUTION;

EID: 0030568611     PISSN: 00142999     EISSN: None     Source Type: Journal    
DOI: 10.1016/0014-2999(96)00279-8     Document Type: Article

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