Preparation of iodine-123 labeled AM251: A potential spect radioligand for the brain cannabinoid CB1 receptor

Journal of Labelled Compounds and Radiopharmaceuticals

Volumn 38, Issue 10, 1996, Pages 875-881

  Lan, Ruoxi ^a   Gatley, S John ^b   Makriyannis, Alexandros ^a  

^a UNIVERSITY OF CONNECTICUT   (United States)

^b BROOKHAVEN NATIONAL LABORATORY   (United States)

Author keywords

Cannabinoid receptor antagonist; Iodine 123; SR141617A

Indexed keywords

1H-PYRAZOLE; 4-IODOPHENYL; CANNABINOID RECEPTOR ANTAGONIST; CANNABINOID RECEPTORS; CANNABINOIDS; IODINE-123; LABELINGS; RADIOLIGANDS; RECEPTOR ANTAGONISTS; SR141617A;

IODINE;

1 (2,4 DICHLOROPHENYL) 5 (4 IODOPHENYL) 4 METHYL N (1 PIPERIDYL) 1H PYRAZOLE 3 CARBOXAMIDE; CANNABINOID RECEPTOR; IODINE 123; RADIOLIGAND; RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ANIMAL EXPERIMENT; ARTICLE; BRAIN LEVEL; DRUG DISTRIBUTION; DRUG SYNTHESIS; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; INTRAVENOUS DRUG ADMINISTRATION; ISOTOPE LABELING; MOUSE; NONHUMAN; REACTION ANALYSIS; ULTRAVIOLET SPECTROPHOTOMETRY;

ANIMALIA;

EID: 0029798021     PISSN: 03624803     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1099-1344(199610)38:10<875::AID-JLCR908>3.0.CO;2-G     Document Type: Article

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