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ChemMedChem

Volumn 1, Issue 9, 2006, Pages 959-964

Correlation of biological activity with active site binding modes of geminal disulfone HIV-1 integrase inhibitors

(3) Meadows, D Christopher a Tantillo, Dean J a Gervay Hague, Jacquelyn a

a UNIVERSITY OF CALIFORNIA (United States)

Author keywords

AutoDock; Binding modes; HIV; Inhibitors; Integrase

Indexed keywords

INTEGRASE; INTEGRASE INHIBITOR; SULFONE;

ANIMAL; ARTICLE; BINDING SITE; CATALYSIS; CHEMICAL STRUCTURE; CHEMISTRY; DRUG EFFECT; ENZYMOLOGY; HUMAN; HUMAN IMMUNODEFICIENCY VIRUS 1; HYDROGEN BOND; METABOLISM; SYNTHESIS;

ANIMALS; BINDING SITES; CATALYSIS; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; HIV-1; HUMANS; HYDROGEN BONDING; MODELS, MOLECULAR; SULFONES;

EID: 33749016010 PISSN: 18607179 EISSN: 18607187 Source Type: Journal
DOI: 10.1002/cmdc.200600040 Document Type: Article

Times cited : (6)

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