Discovery of a Novel Binding Trench in HIV Integrase

Journal of Medicinal Chemistry

Volumn 47, Issue 8, 2004, Pages 1879-1881

  Schames, Julie R ^a   Henchman, Richard H ^a   Siegel, Jay S ^a   Sotriffer, Christoph A ^a   Ni, Haihong ^a   McCammon, J Andrew ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

INTEGRASE; VIRUS DNA;

ARTICLE; BINDING SITE; COMPLEX FORMATION; CRYSTAL STRUCTURE; DNA INTEGRATION; DRUG BINDING; ENZYME ACTIVE SITE; HUMAN IMMUNODEFICIENCY VIRUS 1; HUMAN IMMUNODEFICIENCY VIRUS INFECTION; MOLECULAR DYNAMICS; PROTEIN STRUCTURE; X RAY ANALYSIS;

BINDING SITES; CRYSTALLOGRAPHY, X-RAY; HIV INTEGRASE; INDOLES; LIGANDS; MODELS, MOLECULAR; MOLECULAR CONFORMATION; NAPHTHALENES; PROTEIN BINDING; STRUCTURE-ACTIVITY RELATIONSHIP; TETRAZOLES;

EID: 1842607357     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0341913     Document Type: Article

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