-
1
-
-
1642302295
-
Experience with therapeutic drug monitoring of cyclosporine
-
Abendroth D. Experience with therapeutic drug monitoring of cyclosporine. Transplant Proc 2004; 36: 426S-29S.
-
(2004)
Transplant Proc
, vol.36
-
-
Abendroth, D.1
-
3
-
-
0343416856
-
Contributions of hepatic and intestinal metabolism and P-glycoprotein to cyclosporine and tacrolimus oral drug delivery
-
Hebert MF. Contributions of hepatic and intestinal metabolism and P-glycoprotein to cyclosporine and tacrolimus oral drug delivery. Adv Drug Deliv Rev 1997; 27: 201-14.
-
(1997)
Adv Drug Deliv Rev
, vol.27
, pp. 201-214
-
-
Hebert, M.F.1
-
4
-
-
0028825399
-
Absence of the mdr1a P-Glycoprotein in mice affects tissue distribution and pharmacokinetics of dexamethasone, digoxin, and cyclosporin A
-
Schinkel AH, Wagenaar E, van Deemter L, Mol CA, Borst P. Absence of the mdr1a P-Glycoprotein in mice affects tissue distribution and pharmacokinetics of dexamethasone, digoxin, and cyclosporin A. J Clin Invest 1995; 96: 1698-705.
-
(1995)
J Clin Invest
, vol.96
, pp. 1698-1705
-
-
Schinkel, A.H.1
Wagenaar, E.2
Van Deemter, L.3
Mol, C.A.4
Borst, P.5
-
5
-
-
2442700486
-
Drug-drug, drug-dietary supplement and drug-citrus fruit and other food interactions: What have we learned?
-
Huang SM, Lesko LJ. Drug-drug, drug-dietary supplement and drug-citrus fruit and other food interactions: what have we learned? J Clin Pharmacol 2004; 44: 559-69.
-
(2004)
J Clin Pharmacol
, vol.44
, pp. 559-569
-
-
Huang, S.M.1
Lesko, L.J.2
-
6
-
-
0030982634
-
Grapefruit juice increases felodipine oral availability in humans by decreasing intestinal CYP3A protein expression
-
Lown KS, Bailey DG, Fontana RJ, Janardan SK, Adair CH, Fortlage LA, Brown MB, Guo W, Watkins PB. Grapefruit juice increases felodipine oral availability in humans by decreasing intestinal CYP3A protein expression. J Clin Invest 1997; 99: 2545-53.
-
(1997)
J Clin Invest
, vol.99
, pp. 2545-2553
-
-
Lown, K.S.1
Bailey, D.G.2
Fontana, R.J.3
Janardan, S.K.4
Adair, C.H.5
Fortlage, L.A.6
Brown, M.B.7
Guo, W.8
Watkins, P.B.9
-
7
-
-
14344258321
-
Two major grapefruit juice components differ in time to onset of intestinal CYP3A4 inhibition
-
Paine MF, Criss AB, Watkins PB. Two major grapefruit juice components differ in time to onset of intestinal CYP3A4 inhibition. J Pharmacol Exp Ther 2005; 312: 1151-60.
-
(2005)
J Pharmacol Exp Ther
, vol.312
, pp. 1151-1160
-
-
Paine, M.F.1
Criss, A.B.2
Watkins, P.B.3
-
8
-
-
16244386204
-
Probable interaction of bergamottin and cyclosporine in a lung transplant recipient
-
Johnston PE, Milstone A. Probable interaction of bergamottin and cyclosporine in a lung transplant recipient. Transplantation 2005; 79: 746.
-
(2005)
Transplantation
, vol.79
, pp. 746
-
-
Johnston, P.E.1
Milstone, A.2
-
9
-
-
0034640316
-
Amounts and variation in grapefruit juice of the main components causing grapefruit-drug interaction
-
Fukuda K, Guo L, Ohashi N, Yoshikawa M, Yamazoe Y. Amounts and variation in grapefruit juice of the main components causing grapefruit-drug interaction. J Chromatogr B Biomed Sci Appl 2000; 741: 195-203.
-
(2000)
J Chromatogr B Biomed Sci Appl
, vol.741
, pp. 195-203
-
-
Fukuda, K.1
Guo, L.2
Ohashi, N.3
Yoshikawa, M.4
Yamazoe, Y.5
-
10
-
-
0033713294
-
Grapefruit-felodipine interaction: Effect of unprocessed fruit and probable active ingredients
-
Bailey DG, Dresser GK, Kreeft JH, Munoz C, Freeman DJ, Bend JR. Grapefruit-felodipine interaction: effect of unprocessed fruit and probable active ingredients. Clin Pharmacol Ther 2000; 68: 468-77.
-
(2000)
Clin Pharmacol Ther
, vol.68
, pp. 468-477
-
-
Bailey, D.G.1
Dresser, G.K.2
Kreeft, J.H.3
Munoz, C.4
Freeman, D.J.5
Bend, J.R.6
-
11
-
-
0036159433
-
Fruit juices inhibit organic anion transporting polypeptide-mediated drug uptake to decrease the oral availability of fexofenadine
-
Dresser GK, Bailey DG, Leake BF, Schwarz UI, Dawson PA, Freeman DJ, Kim RB. Fruit juices inhibit organic anion transporting polypeptide-mediated drug uptake to decrease the oral availability of fexofenadine. Clin Pharmacol Ther 2002; 71: 11-20.
-
(2002)
Clin Pharmacol Ther
, vol.71
, pp. 11-20
-
-
Dresser, G.K.1
Bailey, D.G.2
Leake, B.F.3
Schwarz, U.I.4
Dawson, P.A.5
Freeman, D.J.6
Kim, R.B.7
-
12
-
-
0031445547
-
Characterization of interintestinal and intraintestinal variations in human CYP3A-dependent metabolism
-
Paine MF, Khalighi M, Fisher JM, Shen DD, Kunze KL, Marsh CL, Perkins JD, Thummel KE. Characterization of interintestinal and intraintestinal variations in human CYP3A-dependent metabolism. J Pharmacol Exp Ther 1997; 283: 1552-62.
-
(1997)
J Pharmacol Exp Ther
, vol.283
, pp. 1552-1562
-
-
Paine, M.F.1
Khalighi, M.2
Fisher, J.M.3
Shen, D.D.4
Kunze, K.L.5
Marsh, C.L.6
Perkins, J.D.7
Thummel, K.E.8
-
13
-
-
12644272784
-
Role of intestinal P-glycoprotein (mdr1) in interpatient variation in the oral bioavailability of cyclosporine
-
Lown KS, Mayo RR, Leichtman AB, Hsiao HL, Turgeon DK, Schmiedlin-Ren P, Brown MB, Guo W, Rossi SJ, Benet LZ, Watkins PB. Role of intestinal P-glycoprotein (mdr1) in interpatient variation in the oral bioavailability of cyclosporine. Clin Pharmacol Ther 1997; 62: 248-60.
-
(1997)
Clin Pharmacol Ther
, vol.62
, pp. 248-260
-
-
Lown, K.S.1
Mayo, R.R.2
Leichtman, A.B.3
Hsiao, H.L.4
Turgeon, D.K.5
Schmiedlin-Ren, P.6
Brown, M.B.7
Guo, W.8
Rossi, S.J.9
Benet, L.Z.10
Watkins, P.B.11
-
14
-
-
4344656740
-
CYP3A4 and P-glycoprotein activity in healthy controls and transplant patients on cyclosporin vs. tacrolimus vs. sirolimus
-
Lemahieu WP, Maes BD, Verbeke K, Vanrenterghem Y. CYP3A4 and P-glycoprotein activity in healthy controls and transplant patients on cyclosporin vs. tacrolimus vs. sirolimus. Am J Transplant 2004; 4: 1514-22.
-
(2004)
Am J Transplant
, vol.4
, pp. 1514-1522
-
-
Lemahieu, W.P.1
Maes, B.D.2
Verbeke, K.3
Vanrenterghem, Y.4
-
16
-
-
0037766006
-
Association of the CYP3A4*1B 5′-flanking region polymorphism with cyclosporine pharmacokinetics in healthy subjects
-
Min DI, Ellingrod VL. Association of the CYP3A4*1B 5′-flanking region polymorphism with cyclosporine pharmacokinetics in healthy subjects. Ther Drug Monit 2003; 25: 305-9.
-
(2003)
Ther Drug Monit
, vol.25
, pp. 305-309
-
-
Min, D.I.1
Ellingrod, V.L.2
-
17
-
-
10044294681
-
Population pharmacokinetics of cyclosporine in kidney and heart transplant recipients and the influence of ethnicity and genetic polymorphisms in the MDR-1, CYP3A4, and CYP3A5 genes
-
Hesselink DA, van Gelder T, van Schaik RH, Balk AH, van der Heiden IP, van Dam T, van der Werf M, Weimar W, Mathot RA. Population pharmacokinetics of cyclosporine in kidney and heart transplant recipients and the influence of ethnicity and genetic polymorphisms in the MDR-1, CYP3A4, and CYP3A5 genes. Clin Pharmacol Ther 2004; 76: 545-56.
-
(2004)
Clin Pharmacol Ther
, vol.76
, pp. 545-556
-
-
Hesselink, D.A.1
Van Gelder, T.2
Van Schaik, R.H.3
Balk, A.H.4
Van Der Heiden, I.P.5
Van Dam, T.6
Van Der Werf, M.7
Weimar, W.8
Mathot, R.A.9
-
18
-
-
13144282667
-
Association of CYP3A4 genotype with treatment-related leukemia
-
Felix CA, Walker AH, Lange BJ, Williams TM, Winick NJ, Cheung NK, Lovett BD, Nowell PC, Blair IA, Rebbeck TR. Association of CYP3A4 genotype with treatment-related leukemia. Proc Natl Acad Sci USA 1998; 95: 13176-81.
-
(1998)
Proc Natl Acad Sci USA
, vol.95
, pp. 13176-13181
-
-
Felix, C.A.1
Walker, A.H.2
Lange, B.J.3
Williams, T.M.4
Winick, N.J.5
Cheung, N.K.6
Lovett, B.D.7
Nowell, P.C.8
Blair, I.A.9
Rebbeck, T.R.10
-
19
-
-
0041831261
-
Genetic polymorphisms of the CYP3A4, CYP3A5, and MDR-1 genes and pharmacokinetics of the calcineurin inhibitors cyclosporine and tacrolimus
-
Hesselink DA, van Schaik RH, van der Heiden IP, van der Werf M, Gregoor PJ, Lindemans J, Weimar W, van Gelder T. Genetic polymorphisms of the CYP3A4, CYP3A5, and MDR-1 genes and pharmacokinetics of the calcineurin inhibitors cyclosporine and tacrolimus. Clin Pharmacol Ther 2003; 74: 245-54.
-
(2003)
Clin Pharmacol Ther
, vol.74
, pp. 245-254
-
-
Hesselink, D.A.1
Van Schaik, R.H.2
Van Der Heiden, I.P.3
Van Der Werf, M.4
Gregoor, P.J.5
Lindemans, J.6
Weimar, W.7
Van Gelder, T.8
-
20
-
-
0034744113
-
No influence of the MDR-1 C3435T polymorphism or a CYP3A4 promoter polymorphism (CYP3A4-V allele) on dose-adjusted cyclosporin a trough concentrations or rejection incidence in stable renal transplant recipients
-
von Ahsen N, Richter M, Grupp C, Ringe B, Oellerich M, Armstrong VW. No influence of the MDR-1 C3435T polymorphism or a CYP3A4 promoter polymorphism (CYP3A4-V allele) on dose-adjusted cyclosporin A trough concentrations or rejection incidence in stable renal transplant recipients. Clin Chem 2001; 47: 1048-52.
-
(2001)
Clin Chem
, vol.47
, pp. 1048-1052
-
-
Von Ahsen, N.1
Richter, M.2
Grupp, C.3
Ringe, B.4
Oellerich, M.5
Armstrong, V.W.6
-
21
-
-
12144286933
-
The effect of CYP3A5 and MDR1 (ABCB1) polymorphisms on cyclosporine and tacrolimus dose requirements and trough blood levels in stable renal transplant patients
-
Haufroid V, Mourad M, Van Kerckhove V, Wawrzyniak J, De Meyer M, Eddour DC, Malaise J, Lison D, Squifflet JP, Wallemacq P. The effect of CYP3A5 and MDR1 (ABCB1) polymorphisms on cyclosporine and tacrolimus dose requirements and trough blood levels in stable renal transplant patients. Pharmacogenetics 2004; 14: 147-54.
-
(2004)
Pharmacogenetics
, vol.14
, pp. 147-154
-
-
Haufroid, V.1
Mourad, M.2
Van Kerckhove, V.3
Wawrzyniak, J.4
De Meyer, M.5
Eddour, D.C.6
Malaise, J.7
Lison, D.8
Squifflet, J.P.9
Wallemacq, P.10
-
22
-
-
0036001238
-
C3435T mutation in exon 26 of the human MDR1 gene and cyclosporine pharmacokinetics in healthy subjects
-
Min DI, Ellingrod VL. C3435T mutation in exon 26 of the human MDR1 gene and cyclosporine pharmacokinetics in healthy subjects. Ther Drug Monit 2002; 24: 400-4.
-
(2002)
Ther Drug Monit
, vol.24
, pp. 400-404
-
-
Min, D.I.1
Ellingrod, V.L.2
-
23
-
-
1642523162
-
Polymorphisms in human MDR1 (P-glycoprotein): Recent advances and clinical relevance
-
Marzolini C, Paus E, Buclin T, Kim RB. Polymorphisms in human MDR1 (P-glycoprotein): recent advances and clinical relevance. Clin Pharmacol Ther 2004; 75: 13-33.
-
(2004)
Clin Pharmacol Ther
, vol.75
, pp. 13-33
-
-
Marzolini, C.1
Paus, E.2
Buclin, T.3
Kim, R.B.4
-
24
-
-
0033996319
-
Content of CYP3A4 inhibitors, naringin, naringenin and bergapten in grapefruit and grapefruit juice products
-
Ho PC, Saville DJ, Coville PF, Wanwimolruk S. Content of CYP3A4 inhibitors, naringin, naringenin and bergapten in grapefruit and grapefruit juice products. Pharm Acta Helv 2000; 74: 379-85.
-
(2000)
Pharm Acta Helv
, vol.74
, pp. 379-385
-
-
Ho, P.C.1
Saville, D.J.2
Coville, P.F.3
Wanwimolruk, S.4
-
25
-
-
0342868292
-
Role of furanocoumarin derivatives on grapefruit juice-mediated inhibition of human CYP3A activity
-
Guo LQ, Fukuda K, Ohta T, Yamazoe Y. Role of furanocoumarin derivatives on grapefruit juice-mediated inhibition of human CYP3A activity. Drug Metab Dispos 2000; 28: 766-71.
-
(2000)
Drug Metab Dispos
, vol.28
, pp. 766-771
-
-
Guo, L.Q.1
Fukuda, K.2
Ohta, T.3
Yamazoe, Y.4
-
26
-
-
0242469224
-
The effects of fruit juices on drug disposition: A new model for drug interactions
-
Dresser GK, Bailey DG. The effects of fruit juices on drug disposition: a new model for drug interactions. Eur J Clin Invest 2003; 33 (Suppl. 2): 10-6.
-
(2003)
Eur J Clin Invest
, vol.33
, Issue.2 SUPPL.
, pp. 10-16
-
-
Dresser, G.K.1
Bailey, D.G.2
-
27
-
-
4644267926
-
Two major grapefruit juice components differ in intestinal CYP3A4 inhibition kinetic and binding properties
-
Paine MF, Criss AB, Watkins PB. Two major grapefruit juice components differ in intestinal CYP3A4 inhibition kinetic and binding properties. Drug Metab Dispos 2004; 32: 1146-53.
-
(2004)
Drug Metab Dispos
, vol.32
, pp. 1146-1153
-
-
Paine, M.F.1
Criss, A.B.2
Watkins, P.B.3
-
28
-
-
0028963036
-
Effect of grapefruit juice on blood cyclosporin concentration
-
Yee GC, Stanley DL, Pessa LJ, Dalla Costa T, Beltz SE, Ruiz J, Lowenthal DT. Effect of grapefruit juice on blood cyclosporin concentration. Lancet 1995; 345: 955-6.
-
(1995)
Lancet
, vol.345
, pp. 955-956
-
-
Yee, G.C.1
Stanley, D.L.2
Pessa, L.J.3
Dalla Costa, T.4
Beltz, S.E.5
Ruiz, J.6
Lowenthal, D.T.7
-
29
-
-
0031784578
-
Effect of grapefruit juice on the pharmacokinetics of microemulsion cyclosporine and its metabolite in healthy volunteers: Does the formulation difference matter?
-
Ku YM, Min DI, Flanigan M. Effect of grapefruit juice on the pharmacokinetics of microemulsion cyclosporine and its metabolite in healthy volunteers: does the formulation difference matter? J Clin Pharmacol 1998; 38: 959-65.
-
(1998)
J Clin Pharmacol
, vol.38
, pp. 959-965
-
-
Ku, Y.M.1
Min, D.I.2
Flanigan, M.3
-
30
-
-
0035126980
-
Effect of grapefruit juice on pharmacokinetics of microemulsion cyclosporine in African American subjects compared with Caucasian subjects: Does ethnic difference matter?
-
Lee M, Min DI, Ku YM, Flanigan M. Effect of grapefruit juice on pharmacokinetics of microemulsion cyclosporine in African American subjects compared with Caucasian subjects: does ethnic difference matter? J Clin Pharmacol 2001; 41: 317-23.
-
(2001)
J Clin Pharmacol
, vol.41
, pp. 317-323
-
-
Lee, M.1
Min, D.I.2
Ku, Y.M.3
Flanigan, M.4
-
31
-
-
0035145184
-
Effect of grapefruit juice on Sandimmun Neoral absorption among stable renal allograft recipients
-
Bistrup C, Nielsen FT, Jeppesen UE, Dieperink H. Effect of grapefruit juice on Sandimmun Neoral absorption among stable renal allograft recipients. Nephrol Dial Transplant 2001; 16: 373-7.
-
(2001)
Nephrol Dial Transplant
, vol.16
, pp. 373-377
-
-
Bistrup, C.1
Nielsen, F.T.2
Jeppesen, U.E.3
Dieperink, H.4
-
32
-
-
0029890499
-
Effect of grapefruit juice on cyclosporine pharmacokinetics in renal transplant patients
-
Min DI, Ku YM, Perry PJ, Ukah FO, Ashton K, Martin MF, Hunsicker LG. Effect of grapefruit juice on cyclosporine pharmacokinetics in renal transplant patients. Transplantation 1996; 62: 123-5.
-
(1996)
Transplantation
, vol.62
, pp. 123-125
-
-
Min, D.I.1
Ku, Y.M.2
Perry, P.J.3
Ukah, F.O.4
Ashton, K.5
Martin, M.F.6
Hunsicker, L.G.7
-
33
-
-
10044240240
-
Bergamottin contribution to the grapefruit juice-felodipine interaction and disposition in humans
-
Goosen TC, Cillie D, Bailey DG, Yu C, He K, Hollenberg PF, Woster PM, Cohen L, Williams JA, Rheeders M, Dijkstra HP. Bergamottin contribution to the grapefruit juice-felodipine interaction and disposition in humans. Clin Pharmacol Ther 2004; 76: 607-17.
-
(2004)
Clin Pharmacol Ther
, vol.76
, pp. 607-617
-
-
Goosen, T.C.1
Cillie, D.2
Bailey, D.G.3
Yu, C.4
He, K.5
Hollenberg, P.F.6
Woster, P.M.7
Cohen, L.8
Williams, J.A.9
Rheeders, M.10
Dijkstra, H.P.11
-
34
-
-
0031711059
-
Grapefruit juice-felodipine interaction: Effect of naringin and 6′,7′-dihydroxybergamottin in humans
-
Bailey DG, Kreeft JH, Munoz C, Freeman DJ, Bend JR. Grapefruit juice-felodipine interaction: effect of naringin and 6′,7′- dihydroxybergamottin in humans. Clin Pharmacol Ther 1998; 64: 248-56.
-
(1998)
Clin Pharmacol Ther
, vol.64
, pp. 248-256
-
-
Bailey, D.G.1
Kreeft, J.H.2
Munoz, C.3
Freeman, D.J.4
Bend, J.R.5
-
35
-
-
0030868487
-
Specific CYP3A4 inhibitors in grapefruit juice: Furocoumarin dimers as components of drug interaction
-
Fukuda K, Ohta T, Oshima Y, Ohashi N, Yoshikawa M, Yamazoe Y. Specific CYP3A4 inhibitors in grapefruit juice: furocoumarin dimers as components of drug interaction. Pharmacogenetics 1997; 7: 391-6.
-
(1997)
Pharmacogenetics
, vol.7
, pp. 391-396
-
-
Fukuda, K.1
Ohta, T.2
Oshima, Y.3
Ohashi, N.4
Yoshikawa, M.5
Yamazoe, Y.6
-
36
-
-
0034660149
-
Inhibition selectivity of grapefruit juice components on human cytochromes P450
-
Tassaneeyakul W, Guo LQ, Fukuda K, Ohta T, Yamazoe Y. Inhibition selectivity of grapefruit juice components on human cytochromes P450. Arch Biochem Biophys 2000; 378: 356-63.
-
(2000)
Arch Biochem Biophys
, vol.378
, pp. 356-363
-
-
Tassaneeyakul, W.1
Guo, L.Q.2
Fukuda, K.3
Ohta, T.4
Yamazoe, Y.5
-
37
-
-
0033913305
-
Effect of furanocoumarin derivatives in grapefruit juice on the uptake of vinblastine by Caco-2 cells and on the activity of cytochrome P450 3A4
-
Ohnishi A, Matsuo H, Yamada S, Takanaga H, Morimoto S, Shoyama Y, Ohtani H, Sawada Y. Effect of furanocoumarin derivatives in grapefruit juice on the uptake of vinblastine by Caco-2 cells and on the activity of cytochrome P450 3A4. Br J Pharmacol 2000; 130: 1369-77.
-
(2000)
Br J Pharmacol
, vol.130
, pp. 1369-1377
-
-
Ohnishi, A.1
Matsuo, H.2
Yamada, S.3
Takanaga, H.4
Morimoto, S.5
Shoyama, Y.6
Ohtani, H.7
Sawada, Y.8
-
38
-
-
0043128579
-
Time course of recovery of cytochrome p450 3A function after single doses of grapefruit juice
-
Greenblatt DJ, von Moltke LL, Harmatz JS, Chen G, Weemhoff JL, Jen C, Kelley CJ, LeDuc BW, Zinny MA. Time course of recovery of cytochrome p450 3A function after single doses of grapefruit juice. Clin Pharmacol Ther 2003; 74: 121-9.
-
(2003)
Clin Pharmacol Ther
, vol.74
, pp. 121-129
-
-
Greenblatt, D.J.1
Von Moltke, L.L.2
Harmatz, J.S.3
Chen, G.4
Weemhoff, J.L.5
Jen, C.6
Kelley, C.J.7
LeDuc, B.W.8
Zinny, M.A.9
-
39
-
-
10844279077
-
Effects of grapefruit juice and orange juice components on P-glycoprotein- and MRP2-mediated drug efflux
-
Honda Y, Ushigome F, Koyabu N, Morimoto S, Shoyama Y, Uchiumi T, Kuwano M, Ohtani H, Sawada Y. Effects of grapefruit juice and orange juice components on P-glycoprotein- and MRP2-mediated drug efflux. Br J Pharmacol 2004; 143: 856-64.
-
(2004)
Br J Pharmacol
, vol.143
, pp. 856-864
-
-
Honda, Y.1
Ushigome, F.2
Koyabu, N.3
Morimoto, S.4
Shoyama, Y.5
Uchiumi, T.6
Kuwano, M.7
Ohtani, H.8
Sawada, Y.9
-
40
-
-
16344378672
-
Grapefruit juice ingestion significantly reduces talinolol bioavailability
-
Schwarz UI, Seemann D, Oertel R, Miehlke S, Kuhlisch E, Fromm MF, Kim RB, Bailey DG, Kirch W. Grapefruit juice ingestion significantly reduces talinolol bioavailability. Clin Pharmacol Ther 2005; 77: 291-301.
-
(2005)
Clin Pharmacol Ther
, vol.77
, pp. 291-301
-
-
Schwarz, U.I.1
Seemann, D.2
Oertel, R.3
Miehlke, S.4
Kuhlisch, E.5
Fromm, M.F.6
Kim, R.B.7
Bailey, D.G.8
Kirch, W.9
|