Melanocortin 4 receptors interact with antimicrobial frog peptide analogues

Biochemical and Biophysical Research Communications

Volumn 343, Issue 4, 2006, Pages 1094-1100

  Do, Ernest U ^a   Jo, Eun Bae ^a   Choi, Gyu ^b   Piao, Long Zhu ^b   Shin, Jaekyoon ^b   Seo, Min Duk ^a   Kang, Su Jin ^a   Lee, Bong Jin ^a   Ho Kim, Kang ^a   Bum Kim, Jae ^a   Kim, Su il ^a  

^a Seoul National University   (South Korea)

^b Sungkyunkwan University   (South Korea)

Author keywords

Agonists and antagonists; Fluorescence polarization; Gaegurin; High throughput screening; Human melanocortin 4 receptors; Rank order of potency

Indexed keywords

5 CARBOXYMETHYLRHODAMINE; ALPHA INTERMEDIN; ALPHA INTERMEDIN DERIVATIVE; ANTIINFECTIVE AGENT; GAEGURIN 5; LUCIFERASE; MELANOCORTIN 4 RECEPTOR; MELANOTAN II; N ACETYL ALPHA INTERMEDIN[4-10]CYCLO[4 NORLEUCINE 5 ASPARTIC ACID 7 [3 (2 NAPHTHYL)ALANINE] 10 LYSINAMIDE]; PEPTIDE DERIVATIVE; PHENYLALANYLLEUCYLGLYCYLALANYLLEUCYLPHENYLALANYLLYSYLTRYPTOPHYLALANYLSERYL LYSINE; PHENYLALANYLLEUCYLGLYCYLLEUCYLPHENYLALANYLLYSYLVALYLALANYLSERYLLYSINE; PHENYLALANYLLEUCYLGLYCYLPHENYLALANYLLEUCYLPHENYLALANYLLEUCYLPHENYLALANYL LYSYLVALYLALANYLSERYLLYSINE; PHENYLALANYLLEUCYLGLYCYLTRYPTOPHYLLEUCYLPHENYLALANYLLYSYLTRYPTOPHYLALANYL SERYLLYSINE; PHENYLALANYLLEUCYLGLYCYLTRYPTOPHYLLEUCYLPHENYLALANYLLYSYLVALYLALANYLSERYL LYSINE; RHODAMINE; TRACER; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG POTENCY; DRUG RECEPTOR BINDING; FLUORESCENCE POLARIZATION IMMUNOASSAY; FROG; IN VITRO STUDY; MEDICINAL PLANT; MICROTITER PLATE ASSAY; NONHUMAN; PRIORITY JOURNAL; REPORTER GENE;

ALPHA-MSH; ANIMALS; ANTIMICROBIAL CATIONIC PEPTIDES; BINDING, COMPETITIVE; CELL LINE; CYCLIC AMP; FLUORESCENCE POLARIZATION; GENES, REPORTER; HUMANS; LIGANDS; MELANOCYTE-STIMULATING HORMONES; OLIGOPEPTIDES; PLANT EXTRACTS; RANIDAE; RECEPTOR, MELANOCORTIN, TYPE 4; RECOMBINANT PROTEINS;

ANURA; RANA RUGOSA;

EID: 33646029969     PISSN: 0006291X     EISSN: 10902104     Source Type: Journal    
DOI: 10.1016/j.bbrc.2006.03.082     Document Type: Article

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