-
1
-
-
0024310869
-
Potent and prolonged acting cyclic lactam analogues of α-melanotropin: Design based on molecular dynamics
-
Al-Obeidi F., Castrucci A. L., Hadley M. E., Hruby V. J. Potent and prolonged acting cyclic lactam analogues of α-melanotropin Design based on molecular dynamics. J. Med. Chem. 32:1989;2555-2561.
-
(1989)
J. Med. Chem.
, vol.32
, pp. 2555-2561
-
-
Al-Obeidi, F.1
Castrucci, A.L.2
Hadley, M.E.3
Hruby, V.J.4
-
4
-
-
0026731363
-
Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA
-
Chhajlani V., Wikberg J. E. S. Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA. FEBS Lett. 309:1992;417-420.
-
(1992)
FEBS Lett.
, vol.309
, pp. 417-420
-
-
Chhajlani, V.1
Wikberg, J.E.S.2
-
5
-
-
0021285596
-
Cyclic melanotropins. 5: Importance of the C-terminal tripeptide (Lys-Pro-Val)
-
Cody W. L., Wilkes B. C., Muska B. J., Hruby V. J., De L. Castrucci A. M., Hadley M. E. Cyclic melanotropins. 5 Importance of the C-terminal tripeptide (Lys-Pro-Val). J. Med. Chem. 27:1984;1186-1190.
-
(1984)
J. Med. Chem.
, vol.27
, pp. 1186-1190
-
-
Cody, W.L.1
Wilkes, B.C.2
Muska, B.J.3
Hruby, V.J.4
De L. Castrucci, A.M.5
Hadley, M.E.6
-
6
-
-
0029980737
-
Evaluation of melanotan-II, a superpotent cyclic melanotropic peptide in a pilot phase-I clinical study
-
Dorr R. T., Lines R., Levine N., Brooks C., Xiang L., Hruby V. J., Hadley M. E. Evaluation of melanotan-II, a superpotent cyclic melanotropic peptide in a pilot phase-I clinical study. Life Sciences. 58:1996;1777-1784.
-
(1996)
Life Sciences.
, vol.58
, pp. 1777-1784
-
-
Dorr, R.T.1
Lines, R.2
Levine, N.3
Brooks, C.4
Xiang, L.5
Hruby, V.J.6
Hadley, M.E.7
-
8
-
-
0027456619
-
Molecular cloning of a novel melanocortin receptor
-
Gantz I., Konda Y., Tashiro T., Shimoto Y., Miwa H., Munzert G., Watson S. J., DelValle J., Yamada T. Molecular cloning of a novel melanocortin receptor. J. Biol. Chem. 268:1993;8246-8250.
-
(1993)
J. Biol. Chem.
, vol.268
, pp. 8246-8250
-
-
Gantz, I.1
Konda, Y.2
Tashiro, T.3
Shimoto, Y.4
Miwa, H.5
Munzert, G.6
Watson, S.J.7
DelValle, J.8
Yamada, T.9
-
9
-
-
0027227288
-
Molecular cloning, expression, and gene localization of a fourth melanocortin receptor
-
Gantz I., Miwa H., Konda Y., Shimoto Y., Tashiro T., Watson S. J., DelValle J., Yamada T. Molecular cloning, expression, and gene localization of a fourth melanocortin receptor. J. Biol. Chem. 268:1993;15174-15179.
-
(1993)
J. Biol. Chem.
, vol.268
, pp. 15174-15179
-
-
Gantz, I.1
Miwa, H.2
Konda, Y.3
Shimoto, Y.4
Tashiro, T.5
Watson, S.J.6
DelValle, J.7
Yamada, T.8
-
11
-
-
0030467905
-
Three dimentional models of the hMC1R melanocortin receptor: Complexes with melanotropin peptide agonists
-
Haskell-Luevano C., Sawyer T. K., Trumpp-Kallmayer S., Bibber J. A., Humlet C., Gantz I., Hruby V. J. Three dimentional models of the hMC1R melanocortin receptor Complexes with melanotropin peptide agonists. Drug Design and Discovery. 14:1996;197-211.
-
(1996)
Drug Design and Discovery
, vol.14
, pp. 197-211
-
-
Haskell-Luevano, C.1
Sawyer, T.K.2
Trumpp-Kallmayer, S.3
Bibber, J.A.4
Humlet, C.5
Gantz, I.6
Hruby, V.J.7
-
12
-
-
0029154516
-
2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin receptors
-
2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin receptors. J. Med. Chem. 38:1995;3454-3461.
-
(1995)
J. Med. Chem.
, vol.38
, pp. 3454-3461
-
-
Hruby, V.J.1
Lu, D.2
Sharma, S.D.3
Castrucci, A.L.4
Kesterson, R.A.5
Al-Obeidi, F.A.6
Hadley, M.E.7
Cone, R.D.8
-
13
-
-
0002293913
-
Melanotropins: Structural, conformational, and biological considerations in the development of superpotent and superprolonged analogs
-
Hruby V. J., Wilkes B. C., Cody W. L., Sawyer T. K., Hadley M. E. Melanotropins Structural, conformational, and biological considerations in the development of superpotent and superprolonged analogs. Peptide Protein Rev. 3:1984;1-64.
-
(1984)
Peptide Protein Rev.
, vol.3
, pp. 1-64
-
-
Hruby, V.J.1
Wilkes, B.C.2
Cody, W.L.3
Sawyer, T.K.4
Hadley, M.E.5
-
14
-
-
0001895147
-
Receptors for the melanocortin peptides in the central nervous system
-
Low, M. J.; Simerly, R. B.; Cone, R. D. Receptors for the melanocortin peptides in the central nervous system. Curr. Opin. Endocr. Diab. 79-88; 1994.
-
(1994)
Curr. Opin. Endocr. Diab.
, pp. 79-88
-
-
Low, M.J.1
Simerly, R.B.2
Cone, R.D.3
-
15
-
-
0026800892
-
The cloning of a family of genes that encode the melanocortin receptors
-
Mountjoy K. G., Robbins L. S., Mortrud M. T., Cone R. D. The cloning of a family of genes that encode the melanocortin receptors. Science. 257:1992;1248-1251.
-
(1992)
Science
, vol.257
, pp. 1248-1251
-
-
Mountjoy, K.G.1
Robbins, L.S.2
Mortrud, M.T.3
Cone, R.D.4
-
16
-
-
0020317281
-
The opiomelanotropinergic neuronal and endocrine systems
-
O'Donahue T. L., Dorsa D. M. The opiomelanotropinergic neuronal and endocrine systems. Peptides. 3:1982;353-395.
-
(1982)
Peptides.
, vol.3
, pp. 353-395
-
-
O'Donahue, T.L.1
Dorsa, D.M.2
-
17
-
-
0029008390
-
A three dimentional model for the interaction of MSH with the melanocortin 1 receptor
-
Prusis P., Frändberg P. A., Muceniece R., Kalvinsh I., Wikberg J. E. S. A three dimentional model for the interaction of MSH with the melanocortin 1 receptor. Biochem. Biophys. Res. Commun. 210:1995;205-210.
-
(1995)
Biochem. Biophys. Res. Commun.
, vol.210
, pp. 205-210
-
-
Prusis, P.1
Frändberg, P.A.2
Muceniece, R.3
Kalvinsh, I.4
Wikberg, J.E.S.5
-
18
-
-
0028104976
-
Synthesis and biological evaluation of α-MSH analogues substituted with alanine
-
Sahm U. G., Oliver G. W. J., Branch S. K., Moss S. H., Pouton C. W. Synthesis and biological evaluation of α-MSH analogues substituted with alanine. Peptides. 15:1994;1297-1302.
-
(1994)
Peptides
, vol.15
, pp. 1297-1302
-
-
Sahm, U.G.1
Oliver, G.W.J.2
Branch, S.K.3
Moss, S.H.4
Pouton, C.W.5
-
19
-
-
0028037667
-
The melanocortin (MC3) receptor from rat hypothalamus: Photoaffinity labelling and binding of alanine-substituted α-MSH analogues
-
Sahm U. G., Qarawi M. A., Oliver G. W. J., Ahmed A. R. H., Branch S. K., Moss S. H., Pouton C. W. The melanocortin (MC3) receptor from rat hypothalamus photoaffinity labelling and binding of alanine-substituted α-MSH analogues. FEBS letters. 350:1994;29-32.
-
(1994)
FEBS Letters
, vol.350
, pp. 29-32
-
-
Sahm, U.G.1
Qarawi, M.A.2
Oliver, G.W.J.3
Ahmed, A.R.H.4
Branch, S.K.5
Moss, S.H.6
Pouton, C.W.7
-
22
-
-
0030564894
-
Major pharmacological distinction of the ACTH receptor from the other melanocortic receptors
-
Schiöth H. B., Chhajlani V., Muceniece R., Klusa V., Wikberg J. E. S. Major pharmacological distinction of the ACTH receptor from the other melanocortic receptors. Life Sciences. 59:1996;797-801.
-
(1996)
Life Sciences
, vol.59
, pp. 797-801
-
-
Schiöth, H.B.1
Chhajlani, V.2
Muceniece, R.3
Klusa, V.4
Wikberg, J.E.S.5
-
23
-
-
0242414867
-
Expression of functional melanocortin 1 receptors in insect cells
-
Schiöth H. B., Kuusinen A., Muceniece R., Szardenings M., Keinänen K., Wikberg J. E. S. Expression of functional melanocortin 1 receptors in insect cells. Biochem. Biophys. Res. Commun. 221:1996;807-814.
-
(1996)
Biochem. Biophys. Res. Commun.
, vol.221
, pp. 807-814
-
-
Schiöth, H.B.1
Kuusinen, A.2
Muceniece, R.3
Szardenings, M.4
Keinänen, K.5
Wikberg, J.E.S.6
-
24
-
-
0029961314
-
Characterisation of melanocortin 4 receptor by radioligand binding analysis
-
Schiöth H. B., Muceniece R., Wikberg J. E. S. Characterisation of melanocortin 4 receptor by radioligand binding analysis. Pharmacol. Toxicol. 79:1996;161-165.
-
(1996)
Pharmacol. Toxicol.
, vol.79
, pp. 161-165
-
-
Schiöth, H.B.1
Muceniece, R.2
Wikberg, J.E.S.3
-
26
-
-
0023868553
-
Regulation of the synthesis of steroidogenic enzymes in adrenal cortical cells by ACTH
-
Simpson E. R., Waterman M. R. Regulation of the synthesis of steroidogenic enzymes in adrenal cortical cells by ACTH. Ann. Rev. Physiol. 50:1988;427-440.
-
(1988)
Ann. Rev. Physiol.
, vol.50
, pp. 427-440
-
-
Simpson, E.R.1
Waterman, M.R.2
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