메뉴 건너뛰기




Volumn 18, Issue 7, 1997, Pages 1009-1013

Selectivity of cyclic [D-Nal7] and [D-Phe7] substituted MSH analogues for the melanocortin receptor subtypes

Author keywords

HS9510; Ligand binding; Melanocortin receptor subtypes; MSH; MTII; SHU9119

Indexed keywords

INTERMEDIN DERIVATIVE; RECEPTOR SUBTYPE;

EID: 0030663516     PISSN: 01969781     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0196-9781(97)00079-X     Document Type: Article
Times cited : (84)

References (26)
  • 1
    • 0024310869 scopus 로고
    • Potent and prolonged acting cyclic lactam analogues of α-melanotropin: Design based on molecular dynamics
    • Al-Obeidi F., Castrucci A. L., Hadley M. E., Hruby V. J. Potent and prolonged acting cyclic lactam analogues of α-melanotropin Design based on molecular dynamics. J. Med. Chem. 32:1989;2555-2561.
    • (1989) J. Med. Chem. , vol.32 , pp. 2555-2561
    • Al-Obeidi, F.1    Castrucci, A.L.2    Hadley, M.E.3    Hruby, V.J.4
  • 4
    • 0026731363 scopus 로고
    • Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA
    • Chhajlani V., Wikberg J. E. S. Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA. FEBS Lett. 309:1992;417-420.
    • (1992) FEBS Lett. , vol.309 , pp. 417-420
    • Chhajlani, V.1    Wikberg, J.E.S.2
  • 6
    • 0029980737 scopus 로고    scopus 로고
    • Evaluation of melanotan-II, a superpotent cyclic melanotropic peptide in a pilot phase-I clinical study
    • Dorr R. T., Lines R., Levine N., Brooks C., Xiang L., Hruby V. J., Hadley M. E. Evaluation of melanotan-II, a superpotent cyclic melanotropic peptide in a pilot phase-I clinical study. Life Sciences. 58:1996;1777-1784.
    • (1996) Life Sciences. , vol.58 , pp. 1777-1784
    • Dorr, R.T.1    Lines, R.2    Levine, N.3    Brooks, C.4    Xiang, L.5    Hruby, V.J.6    Hadley, M.E.7
  • 13
    • 0002293913 scopus 로고
    • Melanotropins: Structural, conformational, and biological considerations in the development of superpotent and superprolonged analogs
    • Hruby V. J., Wilkes B. C., Cody W. L., Sawyer T. K., Hadley M. E. Melanotropins Structural, conformational, and biological considerations in the development of superpotent and superprolonged analogs. Peptide Protein Rev. 3:1984;1-64.
    • (1984) Peptide Protein Rev. , vol.3 , pp. 1-64
    • Hruby, V.J.1    Wilkes, B.C.2    Cody, W.L.3    Sawyer, T.K.4    Hadley, M.E.5
  • 14
    • 0001895147 scopus 로고
    • Receptors for the melanocortin peptides in the central nervous system
    • Low, M. J.; Simerly, R. B.; Cone, R. D. Receptors for the melanocortin peptides in the central nervous system. Curr. Opin. Endocr. Diab. 79-88; 1994.
    • (1994) Curr. Opin. Endocr. Diab. , pp. 79-88
    • Low, M.J.1    Simerly, R.B.2    Cone, R.D.3
  • 15
    • 0026800892 scopus 로고
    • The cloning of a family of genes that encode the melanocortin receptors
    • Mountjoy K. G., Robbins L. S., Mortrud M. T., Cone R. D. The cloning of a family of genes that encode the melanocortin receptors. Science. 257:1992;1248-1251.
    • (1992) Science , vol.257 , pp. 1248-1251
    • Mountjoy, K.G.1    Robbins, L.S.2    Mortrud, M.T.3    Cone, R.D.4
  • 16
    • 0020317281 scopus 로고
    • The opiomelanotropinergic neuronal and endocrine systems
    • O'Donahue T. L., Dorsa D. M. The opiomelanotropinergic neuronal and endocrine systems. Peptides. 3:1982;353-395.
    • (1982) Peptides. , vol.3 , pp. 353-395
    • O'Donahue, T.L.1    Dorsa, D.M.2
  • 18
    • 0028104976 scopus 로고
    • Synthesis and biological evaluation of α-MSH analogues substituted with alanine
    • Sahm U. G., Oliver G. W. J., Branch S. K., Moss S. H., Pouton C. W. Synthesis and biological evaluation of α-MSH analogues substituted with alanine. Peptides. 15:1994;1297-1302.
    • (1994) Peptides , vol.15 , pp. 1297-1302
    • Sahm, U.G.1    Oliver, G.W.J.2    Branch, S.K.3    Moss, S.H.4    Pouton, C.W.5
  • 19
    • 0028037667 scopus 로고
    • The melanocortin (MC3) receptor from rat hypothalamus: Photoaffinity labelling and binding of alanine-substituted α-MSH analogues
    • Sahm U. G., Qarawi M. A., Oliver G. W. J., Ahmed A. R. H., Branch S. K., Moss S. H., Pouton C. W. The melanocortin (MC3) receptor from rat hypothalamus photoaffinity labelling and binding of alanine-substituted α-MSH analogues. FEBS letters. 350:1994;29-32.
    • (1994) FEBS Letters , vol.350 , pp. 29-32
    • Sahm, U.G.1    Qarawi, M.A.2    Oliver, G.W.J.3    Ahmed, A.R.H.4    Branch, S.K.5    Moss, S.H.6    Pouton, C.W.7
  • 20
    • 0020325969 scopus 로고
    • 10]-α-melanocyte stimulating hormone: A cyclic α-melanotropin exibiting superagonist biological activity
    • 10]-α-melanocyte stimulating hormone A cyclic α-melanotropin exibiting superagonist biological activity. Proc. Natl. Acad. Sci. USA. 79:1982;1751-1755.
    • (1982) Proc. Natl. Acad. Sci. USA , vol.79 , pp. 1751-1755
    • Sawyer, T.K.1    Hruby, V.J.2    Darman, P.S.3    Hadley, M.E.4
  • 22
    • 0030564894 scopus 로고    scopus 로고
    • Major pharmacological distinction of the ACTH receptor from the other melanocortic receptors
    • Schiöth H. B., Chhajlani V., Muceniece R., Klusa V., Wikberg J. E. S. Major pharmacological distinction of the ACTH receptor from the other melanocortic receptors. Life Sciences. 59:1996;797-801.
    • (1996) Life Sciences , vol.59 , pp. 797-801
    • Schiöth, H.B.1    Chhajlani, V.2    Muceniece, R.3    Klusa, V.4    Wikberg, J.E.S.5
  • 24
    • 0029961314 scopus 로고    scopus 로고
    • Characterisation of melanocortin 4 receptor by radioligand binding analysis
    • Schiöth H. B., Muceniece R., Wikberg J. E. S. Characterisation of melanocortin 4 receptor by radioligand binding analysis. Pharmacol. Toxicol. 79:1996;161-165.
    • (1996) Pharmacol. Toxicol. , vol.79 , pp. 161-165
    • Schiöth, H.B.1    Muceniece, R.2    Wikberg, J.E.S.3
  • 26
    • 0023868553 scopus 로고
    • Regulation of the synthesis of steroidogenic enzymes in adrenal cortical cells by ACTH
    • Simpson E. R., Waterman M. R. Regulation of the synthesis of steroidogenic enzymes in adrenal cortical cells by ACTH. Ann. Rev. Physiol. 50:1988;427-440.
    • (1988) Ann. Rev. Physiol. , vol.50 , pp. 427-440
    • Simpson, E.R.1    Waterman, M.R.2


* 이 정보는 Elsevier사의 SCOPUS DB에서 KISTI가 분석하여 추출한 것입니다.