Inhibition mechanism of the recombinant rat P2X2 receptor in glial cells by suramin and TNP-ATP

Biochemistry

Volumn 45, Issue 1, 2006, Pages 224-233

  Trujillo, Cleber A ^a   Nery, Arthur A ^a   Martins, Antonio Henrique B ^b   Majumder, Paromita ^a   Gonzalez, Fernando A ^c   Ulrich, Henning ^a  

^a UNIVERSITY OF SÃO PAULO   (Brazil)

^b FEDERAL UNIVERSITY OF SÃO PAULO   (Brazil)

^c UNIVERSITY OF PUERTO RICO   (Puerto Rico)

Author keywords

[No Author keywords available]

Indexed keywords

ADENOSINETRIPHOSPHATE; BIOASSAY; CELLS; GENETIC ENGINEERING; NEUROLOGY; RADIOTHERAPY;

ANTAGONIST SURAMIN; NONCOMPETITIVE INHIBITION; RECEPTOR INHIBITION; RECOMBINANT RAT;

ENZYME INHIBITION;

ADENOSINE TRIPHOSPHATE; PICRIC ACID; PURINE P2X RECEPTOR; PURINE P2X2 RECEPTOR; RECOMBINANT RECEPTOR; SURAMIN;

ARTICLE; BINDING SITE; CELL COMMUNICATION; CELL STIMULATION; CHANNEL GATING; GENETIC TRANSFECTION; GLIA CELL; HUMAN; HUMAN CELL; KINETICS; LIGAND BINDING; MATHEMATICAL MODEL; MOUSE; NERVOUS SYSTEM; NONHUMAN; PRIORITY JOURNAL; RADIOASSAY; RECEPTOR DOWN REGULATION; RECEPTOR INTRINSIC ACTIVITY;

ADENOSINE TRIPHOSPHATE; ANIMALS; BINDING, COMPETITIVE; CELLS, CULTURED; ELECTROPHYSIOLOGY; KINETICS; NEUROGLIA; RATS; RECEPTORS, PURINERGIC P2; RECOMBINANT PROTEINS; SURAMIN; TRANSFECTION;

EID: 30144445197     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi051517w     Document Type: Article

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