The β subunit increases the ginkgolide B sensitivity of inhibitory glycine receptors

Neuropharmacology

Volumn 49, Issue 6, 2005, Pages 945-951

  Kondratskaya, Elena L ^a,b,c   Betz, Heinrich ^a   Krishtal, Oleg A ^b   Laube, Bodo ^a  

^a MAX PLANCK INSTITUTE FOR BRAIN RESEARCH   (Germany)

^b BOGOMOLETZ INSTITUTE OF PHYSIOLOGY   (Ukraine)

^c RIKEN BRAIN SCIENCE INSTITUTE   (Japan)

Author keywords

Antagonism; Channel block; Ginkgo biloba; GlyR; Picrotoxin; Specificity

Indexed keywords

GINKGO BILOBA EXTRACT; GINKGOLIDE B; GLYCINE; GLYCINE RECEPTOR; OLIGOMER; PROTEIN M2;

ARTICLE; BETA CHAIN; CONTROLLED STUDY; DRUG EFFECT; DRUG INHIBITION; DRUG SENSITIVITY; ELECTROPHYSIOLOGY; GINKGO BILOBA; HUMAN; IC 50; NONHUMAN; OOCYTE; POINT MUTATION; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN EXPRESSION; PROTEIN LOCALIZATION; RECORDING; SYNAPSE; VOLTAGE CLAMP; XENOPUS;

ANIMALS; DITERPENES; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG INTERACTIONS; ELECTRIC STIMULATION; FIBRINOLYTIC AGENTS; GINKGOLIDES; GLYCINE; INHIBITORY CONCENTRATION 50; LACTONES; MEMBRANE POTENTIALS; MICROINJECTIONS; MUTAGENESIS; OOCYTES; PATCH-CLAMP TECHNIQUES; PROTEIN SUBUNITS; RECEPTORS, GLYCINE; RECOMBINANT PROTEINS; XENOPUS;

EID: 26944493388     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2005.07.001     Document Type: Article

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