Identification of selective inhibitors for the glycosyltransferase murg via high-throughput screening

Chemistry and Biology

Volumn 11, Issue 5, 2004, Pages 703-711

  Hu, Yanan ^a   Helm, Jeremiah S ^a   Chen, Lan ^a   Ginsberg, Cindy ^a   Gross, Benjamin ^a   Kraybill, Brian ^a   Tiyanont, Kittichoat ^a   Fang, Xiao ^a   Wu, Tao ^a   Walker, Suzanne ^a  

^a PRINCETON UNIVERSITY   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

ENZYME INHIBITOR; GLYCOSYLTRANSFERASE; LIGAND; N ACETYLGLUCOSAMINYLTRANSFERASE; OUTER MEMBRANE PROTEIN; UDP N ACETYLGLUCOSAMINE N ACETYLMURAMYL (PENTAPEPTIDE)PYROPHOSPHORYL UNDECAPRENOL N ACETYLGLUCOSAMINE TRANSFERASE; UDP-N-ACETYLGLUCOSAMINE-N-ACETYLMURAMYL-(PENTAPEPTIDE)PYROPHOSPHORYL-UNDECAPRENOL N-ACETYLGLUCOSAMINE TRANSFERASE;

ANIMAL; ARTICLE; CHEMISTRY; DRUG ANTAGONISM; DRUG DESIGN; DRUG SCREENING; ENZYMOLOGY; ESCHERICHIA COLI; FLUORESCENCE POLARIZATION; KINETICS; METABOLISM; METHODOLOGY; SYNTHESIS;

ANIMALS; BACTERIAL OUTER MEMBRANE PROTEINS; DRUG DESIGN; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; ESCHERICHIA COLI; FLUORESCENCE POLARIZATION; GLYCOSYLTRANSFERASES; KINETICS; LIGANDS; N-ACETYLGLUCOSAMINYLTRANSFERASES;

ESCHERICHIA COLI;

EID: 2642555622     PISSN: 10745521     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.chembiol.2004.02.024     Document Type: Article

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