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Volumn 6, Issue 7, 2005, Pages 1173-1177

Development and biological evaluation of potent and specific inhibitors of mitotic kinesin Eg5

(7) Gartner, Michael a Sunder Plassmann, Nils a Seiler, Jeanette b Utz, Mathias b Vernos, Isabelle b Surrey, Thomas b Giannis, Athanassios a

a UNIVERSITY OF LEIPZIG (Germany)

b EUROPEAN MOLECULAR BIOLOGY LABORATORY (Germany)

Author keywords

Antitumor agents; Inhibitors; Kinesin; Monastrol; Structure activity relationships

Indexed keywords

ANTINEOPLASTIC AGENT; CK 0106023; DIMETHYLENASTRON; ENASTROL; ENASTRON; HR 22C16; KINESIN; KINESIN 5 INHIBITOR; MONASTROL; MONASTROL DERIVATIVE; S TRITYLCYSTEINE; TERPENDOLE E; UNCLASSIFIED DRUG;

ARTICLE; CONTROLLED STUDY; DRUG POTENCY; DRUG SCREENING; DRUG SYNTHESIS; HUMAN; HUMAN CELL; MITOSIS; PRIORITY JOURNAL;

ANTINEOPLASTIC AGENTS; CELL CULTURE TECHNIQUES; ENZYME INHIBITORS; HELA CELLS; HUMANS; KINESIN; MITOSIS; PYRIMIDINES; STRUCTURE-ACTIVITY RELATIONSHIP; THIONES;

EID: 22144463476 PISSN: 14394227 EISSN: None Source Type: Journal
DOI: 10.1002/cbic.200500005 Document Type: Article

Times cited : (152)

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