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26844502311
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note
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3: C, 71.98; H, 6.33; N, 7.99. Found: C, 72.30; H, 6.52; N, 7.95.
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32
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26844482866
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unpublished results
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4: C, 50.61; H, 4.55; N, 8.34. Found: C, 50.73; H, 4.40; N, 8.36. The relative stereochemistry was confirmed by an X-ray analysis: Belaj, F.; Kappe, C. O. unpublished results.
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39
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2-mediated variation of the Biginelli reaction giving high yields of dihydropyrimidines of type 7: Hu, E. H.; Sidler, D. R.; Dolling, U.-H. J. Org. Chem. 1998, 63, in press. We thank the authors for a preprint of their work.
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