X-ray structure, conformational analysis, enantioseparation, and determination of absolute configuration of the mitotic kinesin Eg5 inhibitor monastrol

Tetrahedron

Volumn 56, Issue 13, 2000, Pages 1859-1862

  Kappe, C Oliver ^a   Shishkin, Oleg V ^b   Uray, Georg ^a   Verdino, Petra ^a  

^a UNIVERSITY OF GRAZ   (Austria)

^b INSTITUTE FOR SINGLE CRYSTALS   (Ukraine)

Author keywords

Biginelli reactions; Circular dichroism; Conformation; Enantiomeric purity

Indexed keywords

ANTIMITOTIC AGENT; KINESIN; MONASTROL; UNCLASSIFIED DRUG;

ARTICLE; CALCULATION; CIRCULAR DICHROISM; DRUG STRUCTURE; ENANTIOMER; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; NUCLEAR MAGNETIC RESONANCE; PRIORITY JOURNAL; STEREOCHEMISTRY; STRUCTURE ANALYSIS; X RAY DIFFRACTION;

EID: 0034708729     PISSN: 00404020     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0040-4020(00)00116-2     Document Type: Article

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