An Efficient Parallel Synthesis of Capsazepine and Capsazepine Analogs

Combinatorial Chemistry and High Throughput Screening

Volumn 7, Issue 2, 2004, Pages 153-161

  Tafesse, Laykea ^a   Kyle, Donald J ^a  

^a Purdue Pharma Discovery Research   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BENZAZEPINE DERIVATIVE; CAPSAZEPINE; VANILLOID RECEPTOR;

ARTICLE; COMBINATORIAL LIBRARY; COMMERCIAL PHENOMENA; DRUG PURIFICATION; DRUG STRUCTURE; DRUG SYNTHESIS; MEDICAL LITERATURE; PRIORITY JOURNAL;

STAPHYLOCOCCUS PHAGE 3A;

EID: 1942423656     PISSN: 13862073     EISSN: None     Source Type: Journal    
DOI: 10.2174/138620704773120838     Document Type: Article

References (22)

1. Benham, C. D.; Davis, J. B.; Randall, A. D. Neuropharmacology, 2002, 42, 873.
2. Caterina, M. J.; Schumacher, M. A.; Tominaga, M.; Rosen T. A.; Levine J. D.; Julius D. Nature, 1997, 389, 816.
3. Hayes, P.; Meadows, H.; Gunthope, M.; Harries, M.; Duckworth, D.; Cairns, W.; Harrison, D.; Clarke, C.; Ellington, K.; Prinjha, R.; Barton, A.; Medhurst, A.; Smith, G.; Topp, S.; Murdock, P.; Sanger, G.; Terrett, J.; Jenkins, O.; Benham, C.; Randall, A.; Gloger, I.; Davis, J. Pain, 2000, 88, 205.
4. Tominaga M.; Caterrina, M.; Malmberg A.; Rosen T.; Gilbert, H.; Skinner, K.; Raumann, B.; Basbaum, A.; Julius, D. Neuron, 1998, 21, 531.
5. Szallasi A.; Blumberg P. M. Pharmacol. Rev., 1999, 51, 159.
6. Carlton, S. M.; Coggeshall, R. E.; Neurosci. Lett., 2001, 210, 53.
7. (a) Hudson, L. J.; Bevan, S.; Wotherspoon, G.; Gentry, C.; Fox A.; Winter, J.; Eur. J. Neurosci., 2001, 13, 2105.
8. (b) Fukuoka, T.; Tokunaga, A.; Tachibana, T.; Dai, Y.; Yamanaka, H.; Noguchi, K. Pain, 2002, 99, 111.
9. Caterina, M. J.; Leffler, A; Malmberg, A. B.; Martin, W. J.; Trafton, J. ; Petersen-Zeitz, K. R.; Koltzenburg, M.; Basbaum, A. I.; Julius D. Science, 2000, 288, 306.
10. Davis, J. B.; Gary, J.; Gunthope, M. J.; Hatcher, J. P.; Davey, P. T.; Overend, P.; Harries, M. H.; Latcham, J.; Claphams, C.; Atkinson, K.; Hughes, S. A.; Rance, K.; Grau, E.; Harper, A. J.; Pugh P. L.; Rogers, D. C.; Bingham, S. ; Randall A.; Sheardown, S. A. Nature, 2000, 405, 183.
11. Valenzano, K. J.; Grant, E. R.; Wu, G.; Hachicha, M.; Schmid, L.; Tafesse, L.; Sun, Q.; Rotshteyn, Y.; Francis, J.; Limberis, J.; Malik, S.; Whittemore, E. R.; Hodges, D. J. Pharmacol. Exp. Ther., 2003, 306, 377.
12. Pomonis, J. D.; Harrison, J. E.; Mark, L.; Whiteside, G. T.; Bristol, D. R.; Valenzano, K. J.; Walker, M. J. K. J. Pharmacol. Exp. Ther., 2003, 306, 387.
13. Walker, K., Urban, L.; Medhurst, S. J., Patel, S.; Panesar, M.; Fox, A. J.; and McIntyre, P. J. Pharmacol. Exp. Ther., 2003, 304, 56.
14. (a) Kelly, S.; Chapman, V. Brain Res., 2002, 935, 103.
15. (b) Sakurada, T.; Matsumura, T.; Moriyama, T.; Sakurada, C.; Ueno, S.; Sakurada, S. Pharmacol Biochem Behav., 2003, 75, 115.
16. (c) Jung, Y., S.; Cho, T. S.; Moon, C. H.; Shin, H.; S. Eur. J. Pharmacol., 1998, 362, 193.
17. Walpole, C. S. J.; Bevan, S.; Bovermann, G.; Boelsterli, J. J.; Breckenridge, R.; Davis J. W.; Hughes, G. A., James, I.; Oberer, L.; Wunter, J. ; Wrigglesworth, R. J. Med. Chem., 1994, 37, 1942.
18. Diego, A. A.; Costa, A.; Mancheno, B.; Najera, C. Tetrahedron, 2001, 53 (13), 4791.
19. Horiguchi, Y.; Saitoh, T.; Terakado, S.; Honda, K.; Kimura, T.; Toda, J. ; Sano, T. Heterocycles, 2001, 54 (2), 967.
20. Lee, J.; and Lee, J. Syn. Comm., 1999, 29 (23), 4127.
21. (a) For review, see Krow, G. R. Tetrahedron, 1981, 37, 1283.
22. (b) Meyers, A. I.; Hutchings, R. H. Tetrahedron, 1993, 49, 1807.