Autoradiographic characterisation of [ 35S]GTPγS binding stimulation mediated by 5-HT 1B receptor in postmortem human brain

Neuropharmacology

Volumn 48, Issue 1, 2005, Pages 25-33

  Mostany, Ricardo ^a   Pazos, Angel ^a   Castro, M Elena ^a  

^a UNIVERSITY OF CANTABRIA   (Spain)

Author keywords

5 HT 1B; 35S GTP S autoradiography; G proteins; Globus pallidus; Putamen; Serotonin; Substantia nigra

Indexed keywords

2,3,6,7 TETRAHYDRO 1' METHYL 5 [[2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL) 4 BIPHENYLYL]CARBONYL]SPIRO[FURO[2,3 F]INDOLE 3,4' PIPERIDINE]; 3 (1,2,5,6 TETRAHYDRO 4 PYRIDYL)PYRROLO[3,2 B]PYRIDIN 5 ONE; 3 [4 (3 CHLOROPHENYL) 1 PIPERAZINYL] 1,1 DIPHENYL 2 PROPANOL; GUANINE NUCLEOTIDE BINDING PROTEIN; GUANOSINE 5' O (3 THIOTRIPHOSPHATE); N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; N [4 METHOXY 3 (4 METHYL 1 PIPERAZINYL)PHENYL] 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL)[1,1' BIPHENYL] 4 CARBOXAMIDE; SEROTONIN; SEROTONIN 1A ANTAGONIST; SEROTONIN 1B ANTAGONIST; SEROTONIN 1B RECEPTOR; SEROTONIN 1D AGONIST; SEROTONIN 1D ANTAGONIST; SEROTONIN 5 O CARBOXYMETHYLGLYCYLTYROSAMINE; UNCLASSIFIED DRUG; 3 (1,2,5,6 TETRAHYDROPYRID 4 YL)PYRROLO(3,2 B)PYRID 5 ONE; 3-(1,2,5,6-TETRAHYDROPYRID-4-YL)PYRROLO(3,2-B)PYRID-5-ONE; BIPHENYL DERIVATIVE; DIPEPTIDE; DRUG DERIVATIVE; OXADIAZOLE DERIVATIVE; PIPERAZINE DERIVATIVE; PIPERIDONE DERIVATIVE; PYRIDINE DERIVATIVE; PYRROLE DERIVATIVE; SB 22489G; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; SEROTONIN O CARBOXYMETHYL GLY TYR; SEROTONIN-O-CARBOXYMETHYL-GLY-TYR; SPIRO COMPOUND; SULFUR;

ADULT; AGED; ARTICLE; AUTOPSY; AUTORADIOGRAPHY; BASAL GANGLION; BRAIN; CAUDATE NUCLEUS; CLINICAL ARTICLE; CONCENTRATION RESPONSE; DENTATE GYRUS; ENTORHINAL CORTEX; FEMALE; GLOBUS PALLIDUS; HIPPOCAMPUS; HUMAN; HUMAN TISSUE; MALE; MESENCEPHALON; PRIORITY JOURNAL; PUTAMEN; SUBSTANTIA NIGRA; BINDING COMPETITION; CADAVER; COMPARATIVE STUDY; DRUG EFFECT; DRUG INTERACTION; HISTOLOGY; METABOLISM; METHODOLOGY; MIDDLE AGED; PROTEIN BINDING;

AGED; AUTORADIOGRAPHY; BINDING, COMPETITIVE; BIPHENYL COMPOUNDS; BRAIN; DIPEPTIDES; DRUG INTERACTIONS; FEMALE; GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE); HUMANS; MALE; MIDDLE AGED; OXADIAZOLES; PIPERAZINES; PIPERIDONES; POSTMORTEM CHANGES; PROTEIN BINDING; PYRIDINES; PYRROLES; RECEPTOR, SEROTONIN, 5-HT1B; SEROTONIN; SEROTONIN AGONISTS; SEROTONIN ANTAGONISTS; SPIRO COMPOUNDS; SULFUR ISOTOPES;

EID: 11144314257     PISSN: 00283908     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.neuropharm.2004.08.013     Document Type: Article

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