Effects of selective h5-HT(1B) (SB-216641) and h5-HT(1D) (BRL-15572) receptor ligands on guinea-pig and human 5-HT auto- and heteroreceptors

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 356, Issue 3, 1997, Pages 321-327

  Schlicker, E ^a   Fink, K ^a   Molderings, G J ^a   Price, G W ^b   Duckworth, M ^b   Gaster, L ^b   Middlemiss, D N ^b   Zentner, J ^a   Likungu, J ^a   Gothert M ^a  

^a UNIVERSITY OF BONN   (Germany)

^b GLAXOSMITHKLINE   (United Kingdom)

Author keywords

BRL 15572; H5 HT(1B) and h5 HT(1D) receptors; Human atrial appendages; Human cerebral cortex; Noradrenaline release; Presynaptic receptors; SB 216641; Serotonin release

Indexed keywords

3 [4 (3 CHLOROPHENYL) 1 PIPERAZINYL] 1,1 DIPHENYL 2 PROPANOL; 5 CARBAMOYLTRYPTAMINE; 6 NITROQUIPAZINE; AUTORECEPTOR; CORTICOSTERONE; DESIPRAMINE; FLUVOXAMINE; IDAZOXAN; METITEPINE; NORADRENALIN; POTASSIUM ION; PRESYNAPTIC RECEPTOR; RECEPTOR SUBTYPE; SB 216641; SEROTONIN; SEROTONIN 1B ANTAGONIST; SEROTONIN 1B RECEPTOR; SEROTONIN 1D ANTAGONIST; SEROTONIN 1D RECEPTOR; SEROTONIN AGONIST; SEROTONIN RECEPTOR AFFECTING AGENT; TRITIUM; UNCLASSIFIED DRUG;

ADOLESCENT; ADULT; ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; BRAIN SLICE; BRAIN SYNAPTOSOME; CONCENTRATION RESPONSE; CONTROLLED STUDY; DRUG SELECTIVITY; ELECTROSTIMULATION; FEMALE; GUINEA PIG; HEART RIGHT ATRIUM; HUMAN; HUMAN TISSUE; MALE; NEUROSURGERY; NEUROTRANSMITTER RELEASE; NONHUMAN; NORADRENALIN RELEASE; SEROTONIN RELEASE;

ANIMALS; AUTORECEPTORS; BENZAMIDES; BIPHENYL COMPOUNDS; CEREBRAL CORTEX; ELECTRIC STIMULATION; GUINEA PIGS; HEART ATRIA; HUMANS; LIGANDS; OXADIAZOLES; PIPERAZINES; POTASSIUM; RECEPTOR, SEROTONIN, 5-HT1B; RECEPTOR, SEROTONIN, 5-HT1D; RECEPTORS, SEROTONIN; SEROTONIN; SEROTONIN ANTAGONISTS; SYNAPTOSOMES; TRITIUM;

EID: 8544222786     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/PL00005057     Document Type: Article

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