Mechanism-Based Approach to the Successful Prevention of Cocaine Inhibition of the Neuronal (α3β4) Nicotinic Acetylcholine Receptor

Biochemistry

Volumn 43, Issue 2, 2004, Pages 481-489

  Krivoshein, Arcadius V ^a   Hess, George P ^a  

^a Department of Obstetrics Gynecology   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CONFORMATIONS; DISSOCIATION; NEUROLOGY; PROTEINS; RNA;

RECEPTOR INHIBITION;

BIOCHEMISTRY;

ACETYLCHOLINE; ALPHA3BETA4 NICOTINIC ACETYLCHOLINE RECEPTOR; ANTICONVULSIVE AGENT; APTAMER; CARBACHOL; CARBOMETHOXYTROPENONE; COCAINE; COCAINE DERIVATIVE; DIZOCILPINE; ECGONINE METHYL ESTER; ION CHANNEL; ISOPROTEIN; LIGAND; NICOTINE; NICOTINIC RECEPTOR; PHENYLTROPANE; PROTEIN INHIBITOR; RECEPTOR SUBTYPE; RNA; UNCLASSIFIED DRUG;

ARTICLE; CELL COMMUNICATION; CHEMICAL REACTION KINETICS; CONCENTRATION (PARAMETERS); CONTROLLED STUDY; DISSOCIATION CONSTANT; DRUG CONFORMATION; DRUG RECEPTOR BINDING; EQUILIBRIUM CONSTANT; HUMAN; HUMAN CELL; INTRACELLULAR RECORDING; ION CURRENT; LIGAND BINDING; MUSCLE; NERVE CELL; NERVOUS SYSTEM; NONHUMAN; PREDICTION; PRIORITY JOURNAL; PROTEIN ANALYSIS; PROTEIN EXPRESSION; RAT; RECEPTOR AFFINITY; RECEPTOR DOWN REGULATION; REGULATORY MECHANISM; SIGNAL TRANSDUCTION;

ANIMALS; BINDING SITES; CARBACHOL; CELL LINE; COCAINE; DIZOCILPINE MALEATE; HUMANS; NEURAL INHIBITION; NEUROMUSCULAR JUNCTION; NICOTINIC AGONISTS; NICOTINIC ANTAGONISTS; PROTEIN CONFORMATION; PROTEIN SUBUNITS; RATS; RECEPTORS, NICOTINIC;

EID: 0347093473     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi034838l     Document Type: Article

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