Reversing the action of noncompetitive inhibitors (MK-801 and cocaine) on a protein (nicotinic acetylcholine receptor)-mediated reaction

Biochemistry

Volumn 42, Issue 20, 2003, Pages 6106-6114

  Hess, George P ^a   Gameiro, Armanda M ^a   Schoenfeld, Ryan C ^b,d   Chen, Yongli ^a   Ulrich, Henning ^a,e   Nye, Jeffrey A ^a,f   Sit, Barbara ^a,g   Carroll, F Ivy ^c   Ganem, Bruce ^b  

^a Department of Obstetrics Gynecology   (United States)

^b Department of Molecular Biology and Genetics   (United States)

^c RTI INTERNATIONAL   (United States)

^d ROCHE BIOSCIENCE   (United States)

^e UNIVERSITY OF SÃO PAULO   (Brazil)

^f UNIVERSITY OF CALIFORNIA   (United States)

^g UNIVERSITY OF WISCONSIN SCHOOL OF MEDICINE AND PUBLIC HEALTH   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CELLS; DERIVATIVES; DRUG DOSAGE; NEUROLOGY; POLYMERIC MEMBRANES; SYNTHESIS (CHEMICAL);

THERAPEUTIC AGENTS;

PROTEINS;

COCAINE; COCAINE DERIVATIVE; DIZOCILPINE; MEMBRANE PROTEIN; NICOTINIC RECEPTOR; NICOTINIC RECEPTOR BLOCKING AGENT; RCS III 140A; RCS III 143; RCS III 202A; RCS III 218; RTI 422970; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; DRUG ABUSE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; MAMMAL; NERVOUS SYSTEM; NONHUMAN; PRIORITY JOURNAL;

ANIMALS; ANTICONVULSANTS; CELL LINE; COCAINE; DIZOCILPINE MALEATE; KINETICS; MAGNETIC RESONANCE SPECTROSCOPY; MICE; MOLECULAR STRUCTURE; NICOTINIC ANTAGONISTS; RECEPTORS, NICOTINIC;

ANIMALIA; MAMMALIA;

EID: 0038521750     PISSN: 00062960     EISSN: None     Source Type: Journal    
DOI: 10.1021/bi020677u     Document Type: Article

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