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Volumn 47, Issue 1, 2004, Pages 262-272

Synthesis and Biological Evaluation of Analogues of 7-Chloro-4,5-dihydro-4-oxo-8-(1,2,4-triazol-4-yl)-1,2,4-triazolo[1,5-a] quinoxaline-2-carboxylic Acid (TQX-173) as Novel Selective AMPA Receptor Antagonists

Author keywords

[No Author keywords available]

Indexed keywords

2 QUINOXALINECARBOXYLIC ACID; 4,5 DIHYDRO 4 OXO 8 (1,2,4 TRIAZOL 4 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; 4,5 DIHYDRO 4 OXO 8 (3 CARBOXYPYRROL 1 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; 4,5 DIHYDRO 4 OXO 8 (3 FORMYLPYRROL 1 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; 4,5 DIHYDRO 4 OXO 8 (PYRROL 1 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; 4,5 DIHYDRO 7 NITRO 4 OXO 8 (3 CARBOXYPYRROL 1 YL) 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLIC ACID; 5,7 DICHLOROKINURENIC ACID; 6 NITRO 7 SULFAMOYLBENZO[F]QUINOXALINE 2,3 DIONE; 7 CHLORO 4,5 DIHYDRO 4 OXO 8 (1,2,4 TRIAZOL 4 YL) 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLIC ACID; ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; AMPA RECEPTOR; AMPA RECEPTOR ANTAGONIST; DIZOCILPINE; ETHYL 4,5 DIHYDRO 4 OXO 8 (1,2,4 TRIAZOL 4 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 4 OXO 8 (3 CARBOXYPYRROL 1 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 4 OXO 8 (3 FORMYL 2,5 DIOXOPYRROL 1 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 4 OXO 8 (3 FORMYLPYRROL 1 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 4 OXO 8 (PYRROL 1 YL) 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 7 NITRO 4 OXO 8 (3 CARBOXYPYRROL 1 YL) 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 7 NITRO 4 OXO 8 (3 FORMYLPYRROL 1 YL) 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 7 NITRO 4 OXO 8 (PYRROL 1 YL) 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 8 (IMIDAZOL 1 YL) 4 OXO 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 4,5 DIHYDRO 8 NITRO 4 OXO 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 8 ACETYLAMINO 4,5 DIHYDRO 7 NITRO 4 OXO 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 8 AMINO 4,5 DIHYDRO 4 OXO 7 TRIFLUOROMETHYL 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; ETHYL 8 AMINO 4,5 DIHYDRO 7 NITRO 4 OXO 1,2,4 TRIAZOLO[1,5 A]QUINOXALINE 2 CARBOXYLATE; FLUORINE DERIVATIVE; ION CHANNEL; KAINIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; TQX 173; UNCLASSIFIED DRUG; UNINDEXED DRUG;

EID: 0346100347     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm030906q     Document Type: Article
Times cited : (46)

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