Synthesis, glycine/NMDA and AMPA binding activity of some new 2,5,6- trioxopyrazino[1,2,3-de]quinoxalines and of their restricted analogs 2,5- dioxo- and 4,5-dioxoimidazo[1,5,4-de]quinoxalines

Archiv der Pharmazie

Volumn 332, Issue 6, 1999, Pages 201-207

  Varano, Flavia ^a   Catarzi, Daniela ^a   Colotta, Vittoria ^a   Cecchi, Lucia ^a   Filacchioni, Guido ^a   Galli, Alessandro ^a   Costagli, Chiara ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

Author keywords

2,5,6 Trioxopyrazino 1,2,3 de quinoxalines; 2,5 dioxoimidazo 1,5,4 de quinoxalines; 4,5 dioxoimidazo 1,5,4 de quinoxalines; Glycine NMDA and AMPA binding activity

Indexed keywords

ALPHA AMINO 3 HYDROXY 5 METHYL 4 ISOXAZOLEPROPIONIC ACID; AMPA RECEPTOR; GLYCINE; N METHYL DEXTRO ASPARTIC ACID; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; QUINOXALINE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; NONHUMAN; PRIORITY JOURNAL; RAT; RECEPTOR AFFINITY; RECEPTOR BINDING; SYNTHESIS;

ANIMALS; MALE; QUINOXALINES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, AMPA; RECEPTORS, GLYCINE; RECEPTORS, N-METHYL-D-ASPARTATE; STRUCTURE-ACTIVITY RELATIONSHIP;

EID: 0033048804     PISSN: 03656233     EISSN: None     Source Type: Journal    
DOI: 10.1002/(SICI)1521-4184(19996)332:6<201::AID-ARDP201>3.0.CO;2-S     Document Type: Article

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