Synthesis of 2-substituted-6,8-dichloro-3,4-dihydro-3-oxo-2H-1,4-benzothiazine-1,1-dioxides and -1-oxides as glycine-NMDA receptor antagonists

Farmaco

Volumn 53, Issue 12, 1998, Pages 752-757

  Varano, Flavia ^a   Catarzi, Daniela ^a   Colotta, Vittoria ^a   Filacchioni, Guido ^a   Cecchi, Lucia ^a   Galli, Alessandro ^a   Costagli, Chiara ^a  

^a UNIVERSITY OF FLORENCE   (Italy)

Author keywords

1,4 Benzothiazine 1,1 dioxides; 1,4 Benzothiazine 1 oxides; Glycine NMDA receptor antagonists

Indexed keywords

1,4 BENZOTHIAZINE 1 OXIDE; 1,4 BENZOTHIAZINE 1,1 DIOXIDE; BENZOTHIAZINE DERIVATIVE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; BINDING AFFINITY; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; MALE; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; RAT; REACTION ANALYSIS;

ANIMALS; BENZOTHIADIAZINES; CEREBRAL CORTEX; EXCITATORY AMINO ACID ANTAGONISTS; MALE; OXIDES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, GLYCINE; RECEPTORS, N-METHYL-D-ASPARTATE; SYNAPTIC MEMBRANES; THIAZINES;

EID: 0032583523     PISSN: 0014827X     EISSN: None     Source Type: Journal    
DOI: 10.1016/S0014-827X(98)00097-4     Document Type: Article

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