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Volumn 22, Issue 7, 2003, Pages 754-766

Solid Phase Combinatorial Library of 1,3-Azole Containing Peptides for the Discovery of Matrix Metallo Proteinase Inhibitors

(4) Christensen, Caspar a Schiødt, Christine Bruun b Foged, Niels Tækker b Meldal, Morten a

a CARLSBERG LABORATORY (Denmark)

b NORDIC BIOSCIENCE A S (Denmark)

Author keywords

Automated bead sorting; Combinatorial chemistry; Dipeptidomimetics; Peptide isosteres; Solid phase peptide chemistry

Indexed keywords

BIOCHIPS; DRUG PRODUCTS; MASS SPECTROMETRY;

AUTOMATED BEAD SORTING; COMBINATORIAL CHEMISTRY; COMBINATORIAL LIBRARY; DIPEPTIDOMIMETIC; PEPTIDE CHEMISTRIES; PEPTIDE ISOSTERE; SOLID PHASE PEPTIDE CHEMISTRY; SOLID PHASIS; SOLID-PHASE; SOLID-PHASE PEPTIDES;

PEPTIDES;

AMINO ACID; MATRIX METALLOPROTEINASE 14; MATRIX METALLOPROTEINASE INHIBITOR; OXAZOLE; PYRROLE DERIVATIVE; THIAZOLE DERIVATIVE;

ARTICLE; COMBINATORIAL LIBRARY; ENZYME ACTIVITY; ENZYME ASSAY; ENZYME KINETICS; MATRIX ASSISTED LASER DESORPTION IONIZATION TIME OF FLIGHT MASS SPECTROMETRY; PRIORITY JOURNAL; SOLID; STATISTICAL ANALYSIS; SYNTHESIS;

EID: 0242551201 PISSN: 1611020X EISSN: None Source Type: Journal
DOI: 10.1002/qsar.200320006 Document Type: Article

Times cited : (17)

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