Steroid Receptor Coactivator Peptidomimetics

Methods in Enzymology

Volumn 364, Issue , 2003, Pages 223-246

  Geistlinger, Timothy R ^a   Guy, R Kiplin ^a  

^a UNIVERSITY OF CALIFORNIA   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CELL NUCLEUS RECEPTOR; ESTROGEN RECEPTOR ALPHA; LACTAM DERIVATIVE; PEPTIDE LIBRARY; PEPTIDOMIMETIC AGENT; STEROID RECEPTOR; SYNTHETIC PEPTIDE; THYROID HORMONE RECEPTOR; UNCLASSIFIED DRUG;

ALPHA HELIX; AMINO ACID SUBSTITUTION; CRYSTAL STRUCTURE; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; FLUORESCENCE POLARIZATION; LIGAND BINDING; PEPTIDE SYNTHESIS; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN FAMILY; PROTEIN PROTEIN INTERACTION; PROTEIN SECONDARY STRUCTURE; REVIEW;

EID: 0242391282     PISSN: 00766879     EISSN: None     Source Type: Book Series    
DOI: 10.1016/S0076-6879(03)64013-9     Document Type: Review

References (41)

1. E. M. McInerney, D. W. Rose, S. E. Flynn, S. Westin, T. M. Mullen, A. Krones, J. Inostroza, J. Torchia, R. T. Nolte, N. Assa-Munt, M. V. Milburn, C. K. Glass, and M. G. Rosenfeld, Genes Dev. 12, 3357-3368 (1998).
2. B. D. Darimont, R. L. Wagner, J. W. Apriletti, M. R. Stallcup, P. J. Kushner, J. D. Baxter, R. J. Fletterick, and K. R. Yamamoto, Genes Dev. 12, 3343-3356 (1998).
3. R. C. Ribeiro, J. W. Apriletti, R. L. Wagner, W. Feng, P. J. Kushner, S. Nilsson, T. S. Scanlan, B. L. West, R. J. Fletterick, and J. D. Baxter, J. Steroid Biochem. Mol. Biol. 65, 133-141 (1998).
4. X. F. Ding, C. M. Anderson, H. Ma, H. Hong, R. M. Uht, P. J. Kushner, and M. R. Stallcup, Mol. Endocrinol. 12, 302-313 (1998).
5. D. M. Heery, E. Kalkhoven, S. Hoare, and M. G. Parker, Nature 387, 733-736 (1997).
6. C. Chang, J. D. Norris, H. Gron, L. A. Paige, P. T. Hamilton, D. J. Kenan, D. Fowlkes, and D. P. McDonnell, Mol. Cell. Biol. 19, 8226-8239 (1999).
7. J. P. Northrop, D. Nguyen, S. Piplani, S. E. Olivan, S. T. Kwan, N. F. Go, C. P. Hart, and P. J. Schatz, Mol. Endocrinol. 14, 605-622 (2000).
8. K. S. Bramllet, Y. Wu, and T. P. Burris, Mol. Endocrinol. 15, 909-922 (2001).
9. M. Needham, S. Raines, J. McPheat, C. Stacey, J. Ellston, S. Hoare, and M. Parker, J. Steroid Biochem. Mol. Biol. 72, 35-46 (2000).
10. J. Zhang and M. A. Lazar, Annu. Rev. Physiol. 62, 439-466 (2000).
11. W. Feng, R. C. Ribeiro, R. L. Wagner, H. Nguyen, J. W. Apriletti, R. J. Fletterick, J. D. Baxter, P. J. Kushner, and B. L. West, Science 280, 1747-1749 (1998).
12. A. K. Shiau, D. Barstad, P. M. Loria, L. Cheng, P. J. Kushner, D. A. Agard, and G. L. Greene, Cell 95, 927-937 (1998).
13. H. E. Xu, M. H. Lambert, V. G. Montana, K. D. Plunket, L. B. Moore, J. L. Collins, J. A. Oplinger, S. A. Kliewer, R. T. Gampe, Jr., D. D. McKee, J. T. Moore, and T. M. Willson, Proc. Natl. Acad. Sci. USA 98, 13919-13924 (2001).
14. R. T. Gampe, Jr., V. G. Montana, M. H. Lambert, G. B. Wisely, M. V. Milburn, and H. E. Xu, Genes Dev. 14, 2229-2241 (2000).
15. R. T. Gampe, Jr., V. G. Montana, M. H. Lambert, A. B. Miller, R. K. Bledsoe, M. V. Milburn, S. A. Kliewer, T. M. Willson, and H. E. Xu, Mol. Cell 5, 545-555 (2000).
16. R. C. Ribeiro, J. W. Apriletti, R. L. Wagner, B. L. West, W. Feng, R. Huber, P. J. Kushner, S. Nilsson, T. Scanlan, R. J. Fletterick, F. Schaufele, and J. D. Baxter, Recent Prog. Horm. Res. 53, 351-392 (1998).
17. Y. Sun, T. J. Ewing, A. G. Skillman, and I. D. Kuntz, J. Comput. Aided Mol. Des. 12, 597-604 (1998).
18. http://www.cgl.ucsf.edu/index.html, U.C.G.L.
19. M. L. Connolly, Science 221, 709-713 (1983).
20. Tripos Associates, I. 1699 South Hanley Road, Suite 303, St. Louis, Missouri 63144-2913, USA.
21. I. D. Kuntz, J. M. Blaney, S. J. Oatley, R. Langridge, and T. E. Ferrin, J. Mol. Biol. 161, 269-288 (1982).
22. R. L. DesJarlais, R. P. Sheridan, G. L. Seibel, J. S. Dixon, I. D. Kuntz, and R. Venkataraghavan, J. Med. Chem. 31, 722-729 (1988).
23. T. J. Ewing, S. Makino, A. G. Skillman, and I. D. Kuntz, J. Comput. Aided Mol. Des. 15, 411-428 (2001).
24. E. C. Meng, B. K. Shoichet, and I. D. Kuntz, J. Comp. Chem. 13, 505-524 (1992).
25. A. G. Skillman, Ph.D. Thesis, UCSF, 1999.
26. 4.6, D.V. Daylight Chemical Information Systems, Inc., Santa Fe, NM, 1997.
27. http://www.daylight.com/dayhtml/doc/theory/theory.finger.html.
28. H. Matter, J. Biolumin. Chemilumin. 40, 1219-1229 (1997).
29. In House Perl Script UCSF.
30. Anchoring - Script, In House Perl Script UCSF.
31. Open Eye Software http://www.eyesopen.com/; J. Boström, J. R. Greenwood, and J. Gottfries, Assessing the performance of OMEGA with respect to retrieving bioactive conformations, J. Mol. Graphics and Modelling 21, 449 (2003).
32. Open Eye Software http://www.eyesopen.com/; J. Boström, J. R. Greenwood, and J. Gottfries, Assessing the performance of OMEGA with respect to retrieving bioactive conformations, J. Mol. Graphics and Modelling 21, 449 (2003).
33. C. Blackburn and S. Kates, Methods Enzymol. 289, 175-198 (1997).
34. T. R. Geistlinger and R. K. Guy, J. Am. Chem. Soc. 123, 1525-1526 (2001).
35. M. Uesugi and G. L. Verdine, Proc. Natl. Acad. Sci. USA 96, 14801-14806 (1999).
36. J. K. Judice, J. Y. Tom, W. Huang, T. Wrin, J. Vennari, C. J. Petropoulos, and R. S. McDowell, Proc. Natl. Acad. Sci. USA 94, 13426-13430 (1997).
37. J. W. Taylor, N. J. Greenfield, B. Wu, and P. L. Privalov, J. Mol. Biol. 291, 965-976 (1999).
38. C. Yu and J. W. Taylor, Bioorg. Med. Chem. 7, 161-175 (1999).
39. T. R. Geistlinger and R. Kiplin Guy, J. Am. Chem. Soc: 125 (23), 6852-6853 (2003).
40. C. Schafmeister, J. Po, and G. Verdine, J. Am. Chem. Soc. 122, 5891-5892 (2000).
41. F. Albericio, P. Lloyd-Williams, and E. Giralt, Methods Enzymol. 289, 313 (1997).