Autoradiographic visualization of corticotropin releasing hormone type 1 receptors with a nonpeptide ligand: Synthesis of [76Br]MJL-1-109-2

Journal of Medicinal Chemistry

Volumn 46, Issue 17, 2003, Pages 3559-3562

  Jagoda, Elaine ^a   Contoreggi, Carlo ^b   Lee, Mei Jing ^c   Kao, Chih Hao K ^a   Szajek, Lawrence P ^a   Listwak, Sam ^d   Gold, Philip ^d   Chrousos, George ^e   Greiner, Elisabeth ^c   Kim, B Moon ^c   Jacobson, Arthur E ^c   Rice, Kenner C ^c   Eckelman, William ^a  

^a NATIONAL INSTITUTES OF HEALTH   (United States)

^b NATIONAL INSTITUTES OF HEALTH   (United States)

^c NATIONAL INSTITUTE OF DIABETES AND DIGESTIVE AND KIDNEY DISEASES   (United States)

^d NATIONAL INSTITUTE OF MENTAL HEALTH   (United States)

^e EUNICE KENNEDY SHRIVER NATIONAL INSTITUTE OF CHILD HEALTH AND HUMAN DEVELOPMENT   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

BUTYL[2,5 DIMETHYL 7 (2,4,6 TRIMETHYLPHENYL) 7H PYRROLO[2,3 D]PYRIMIDIN 4 YL]ETHYLAMINE; CORTICOTROPIN RELEASING FACTOR RECEPTOR; CORTICOTROPIN RELEASING FACTOR RECEPTOR 1; MJL 1 109 2; RADIOLIGAND; TRACER; UNCLASSIFIED DRUG;

ANIMAL TISSUE; ARTICLE; AUTORADIOGRAPHY; BLOOD BRAIN BARRIER; CONTROLLED STUDY; DRUG RECEPTOR BINDING; DRUG STRUCTURE; DRUG SYNTHESIS; LIPOPHILICITY; NONHUMAN; PATHOPHYSIOLOGY; POSITRON EMISSION TOMOGRAPHY; RAT; STRESS;

ANIMALS; AUTORADIOGRAPHY; BLOOD-BRAIN BARRIER; BRAIN; BROMINE RADIOISOTOPES; LIGANDS; RADIOPHARMACEUTICALS; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, CORTICOTROPIN-RELEASING HORMONE; TISSUE DISTRIBUTION; TRIAZINES;

EID: 0042732954     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm034077k     Document Type: Article

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