Studies of the structure of glutamate receptor ion channels and the mechanisms of their blockade by organic cations

Neuroscience and Behavioral Physiology

Volumn 33, Issue 3, 2003, Pages 237-246

  Magazanik, L G ^a   Tikhonov, D B ^a   Bol'shakov, K V ^a   Gmiro, V E ^b   Buldakova, S L ^a   Samoilova, M V ^a  

^a SECHENOV INSTITUTE OF EVOLUTIONARY PHYSIOLOGY AND BIOCHEMISTRY   (Russian Federation)

^b INSTITUTE OF BIOMEDICAL CHEMISTRY   (Russian Federation)

Author keywords

AMPA receptors; Blockers; Glutamate receptors; NMDA receptors

Indexed keywords

1 (1 ADAMANTYLMETHYLAMMONIO) 5 TRIMETHYLAMMONIOPENTANE DIBROMIDE; 1 ADAMANTYLMETHYLAMMONIO 5 AMMONIOPENTANE DIBROMIDE; ADAMANTANE DERIVATIVE; AMANTADINE; AMPA RECEPTOR; AMPA RECEPTOR ANTAGONIST; CATION; GLUTAMATE RECEPTOR; GLYCINE; IEM 1617; IEM 1618; IEM 1921; IEM 2008; IEM 2009; IEM 2010; IEM 2011; IEM 2014; ION CHANNEL; N (5 AMMONIOPENTYL) 1 PHENYLCYCLOHEXYLAMMONIUM DIBROMIDE; N METHYL DEXTRO ASPARTIC ACID RECEPTOR; N METHYL DEXTRO ASPARTIC ACID RECEPTOR BLOCKING AGENT; OXYGEN; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL ISOLATION; CONTROLLED STUDY; DRUG ACTIVITY; DRUG BINDING SITE; DRUG EFFECT; DRUG MECHANISM; DRUG RECEPTOR BINDING; DRUG SELECTIVITY; HYDROPHOBICITY; IC 50; MOLECULAR MECHANICS; MOLECULAR MODEL; NERVE CELL; NONHUMAN; PROTEIN STRUCTURE; RAT; RECEPTOR BLOCKING; STRUCTURE ACTIVITY RELATION; VOLTAGE CLAMP;

ADAMANTANE; AMANTADINE; ANIMALS; ANIMALS, NEWBORN; BRAIN; CATIONS; DOSE-RESPONSE RELATIONSHIP, DRUG; DRUG INTERACTIONS; EXCITATORY AMINO ACID ANTAGONISTS; ION CHANNELS; MODELS, BIOLOGICAL; MODELS, MOLECULAR; NEURONS; PATCH-CLAMP TECHNIQUES; QUATERNARY AMMONIUM COMPOUNDS; RATS; RATS, WISTAR; RECEPTORS, AMPA; RECEPTORS, N-METHYL-D-ASPARTATE;

EID: 0038417896     PISSN: 00970549     EISSN: None     Source Type: Journal    
DOI: 10.1023/A:1022147230445     Document Type: Article

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