Steroid and bile acid conjugates are substrates of human multidrug-resistance protein (MRP) 4 (ATP-binding cassette C4)

Biochemical Journal

Volumn 371, Issue 2, 2003, Pages 361-367

  Zelcer, Noam ^a   Reid, Glen ^a   Wielinga, Peter ^a   Kuil, Annemieke ^a   Van Der Heijden, Ingrid ^a   Schuetz, John D ^b   Borst, Piet ^a  

^a NETHERLANDS CANCER INSTITUTE   (Netherlands)

^b ST JUDE CHILDREN S RESEARCH HOSPITAL   (United States)

Author keywords

Adrenal gland; Bile acid; Cholestasis; Dehydroepiandrosterone 3 sulphate (DHEAS); Multidrug resistance protein (MRP); Steroid

Indexed keywords

CELLS; MEMBRANES; SUBSTRATES;

BILE ACID CONJUGATES;

PROTEINS;

ABC TRANSPORTER; BILE ACID; BILE SALT; CHOLIC ACID; COMPLEMENTARY DNA; CYCLIC AMP; CYCLIC GMP; ESTRADIOL; ESTRADIOL DERIVATIVE; ESTRADIOL DISULFATE; ESTRONE SULFATE; FOLIC ACID; FOLINIC ACID; GLUCURONIDE; GLYCOCHOLIC ACID; GLYCOLITHOCHOLIC ACID; LITHOCHOLIC ACID; METHOTREXATE; MULTIDRUG RESISTANCE PROTEIN 4; PRASTERONE SULFATE; STEROID; SULFATE; TAUROCHENODEOXYCHOLIC ACID; TAUROCHOLIC ACID; TAURODEOXYCHOLIC ACID; TAUROLITHOCHOLATE 3 SULFATE; TAUROLITHOCHOLIC ACID; UNCLASSIFIED DRUG;

ADRENAL GLAND; ARTICLE; CHOLESTASIS; COMPETITIVE INHIBITION; CONTROLLED STUDY; EMBRYO; HUMAN; HUMAN CELL; IMMUNOHISTOCHEMISTRY; KIDNEY CELL; MEMBRANE TRANSPORT; MEMBRANE VESICLE; MULTIDRUG RESISTANCE; PRIORITY JOURNAL; PROTEIN ANALYSIS;

BILE ACIDS AND SALTS; DEHYDROEPIANDROSTERONE SULFATE; DRUG RESISTANCE, MULTIPLE; ESTRADIOL; HUMANS; KINETICS; MULTIDRUG RESISTANCE-ASSOCIATED PROTEINS; RECOMBINANT PROTEINS; STEROIDS; SUBSTRATE SPECIFICITY; TRANSFECTION;

MAMMALIA;

EID: 0037693882     PISSN: 02646021     EISSN: None     Source Type: Journal    
DOI: 10.1042/BJ20021886     Document Type: Article

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