Identification of a peptide antagonist to the peripheral-type benzoidazepine receptor that inhibits hormone-stimulated Leydig cell steroid formation

Journal of Pharmacology and Experimental Therapeutics

Volumn 303, Issue 2, 2002, Pages 627-632

  Gazouli, Maria ^a   Han, Zeqiu ^a   Papadopoulos, Vassilios ^b  

^a GEORGETOWN UNIVERSITY MEDICAL CENTER   (United States)

^b UNIVERSITY OF ATHENS MEDICAL SCHOOL   (Greece)

Author keywords

[No Author keywords available]

Indexed keywords

4' CHLORODIAZEPAM; BENZODIAZEPINE RECEPTOR; BENZODIAZEPINE RECEPTOR BLOCKING AGENT; CHOLESTEROL; CHOLESTEROL DERIVATIVE; CHORIONIC GONADOTROPIN; PERIPHERAL TYPE BENZODIAZEPINE RECEPTOR; SERYLTHREONYLHISTIDYLGLUTAMYLGLUTAMYLHISTIDYLPROLINE; SERYLTHREONYLHISTIDYLGLUTAMYLGLUTAMYLTHREONYLPROLINE; SERYLTHREONYLHISTIDYLGLUTAMYLGLUTAMYLTHREONYLSERINE; SERYLTHREONYLPROLYLHISTIDYLSERYLTHREONYLPROLINE; STEROID; THREONYLALANYLTHREONINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; CELL FUNCTION; CELL STIMULATION; CHOLESTEROL TRANSPORT; DOSE RESPONSE; DRUG COMPETITION; DRUG POTENCY; DRUG RECEPTOR BINDING; HUMAN IMMUNODEFICIENCY VIRUS; IC 50; INHIBITION KINETICS; LEYDIG CELL; LIGAND BINDING; NONHUMAN; PEPTIDE ANALYSIS; PEPTIDE SYNTHESIS; PHAGE DISPLAY; PRIORITY JOURNAL; PROTEIN DOMAIN; PROTEIN MOTIF; RECEPTOR AFFINITY; STEROIDOGENESIS;

ANIMALS; BENZODIAZEPINONES; GENE PRODUCTS, TAT; HORMONES; ISOQUINOLINES; LEYDIG CELL TUMOR; LEYDIG CELLS; LIGANDS; MALE; MICE; MITOCHONDRIA; PEPTIDE FRAGMENTS; PEPTIDE LIBRARY; PERIPHERAL NERVOUS SYSTEM; PROGESTERONE; RECEPTORS, GABA-A; STEROIDS; STRUCTURE-ACTIVITY RELATIONSHIP; THERMODYNAMICS; TUMOR CELLS, CULTURED;

EID: 0036828234     PISSN: 00223565     EISSN: None     Source Type: Journal    
DOI: 10.1124/jpet.102.039388     Document Type: Article

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