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Archives of Biochemistry and Biophysics

Volumn 403, Issue 1, 2002, Pages 41-49

New selective inhibitors of cytochromes P450 2B and their application to antimutagenesis of tamoxifen

(5) Stiborová, Marie a Bořek Dohalská, Lucie a Hodek, Petr a Mráz, Jaroslav b Frei, Eva c

a CHARLES UNIVERSITY (Czech Republic)

b NATIONAL INSTITUTE OF PUBLIC HEALTH (Czech Republic)

c GERMAN CANCER RESEARCH CENTER DKFZ (Germany)

Author keywords

2 isopropenyl 2 methyladamantane; 3 isopropenyl 3 methyldiamantane; Cytochrome P450 2B; DNA adducts; Endometrial cancer; Selective inhibition; Tamoxifen

Indexed keywords

2 ISOPROPENYL 2 METHYLADAMANTANE; 3 ISOPROPENYL 3 METHYLDIAMANTANE; ANTIMUTAGENIC AGENT; CYTOCHROME P450 2B; CYTOCHROME P450 2B INHIBITOR; CYTOCHROME P450 2B2; CYTOCHROME P450 2B4; CYTOCHROME P450 2B6; CYTOCHROME P450 INHIBITOR; TAMOXIFEN; UNCLASSIFIED DRUG;

ARTICLE; CARCINOGENESIS; COMPETITIVE INHIBITION; DNA ADDUCT; DRUG ACTIVATION; DRUG POTENCY; ENDOMETRIUM CANCER; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN; MALE; MICROSOME; NONHUMAN; PRIORITY JOURNAL; RABBIT; RAT;

ADAMANTANE; AMANTADINE; ANIMALS; ANTINEOPLASTIC AGENTS; ARYL HYDROCARBON HYDROXYLASES; CYTOCHROME P-450 ENZYME SYSTEM; DNA ADDUCTS; ENDOMETRIAL NEOPLASMS; ENZYME ACTIVATION; ENZYME INHIBITORS; FEMALE; HUMANS; INHIBITORY CONCENTRATION 50; KINETICS; MICROSOMES; MODELS, CHEMICAL; MUTAGENS; OXYGEN; RABBITS; STEROID HYDROXYLASES; TAMOXIFEN;

ORYCTOLAGUS CUNICULUS;

EID: 0036647214 PISSN: 00039861 EISSN: None Source Type: Journal
DOI: 10.1016/S0003-9861(02)00259-X Document Type: Article

Times cited : (38)

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