Novel inhibitors of poly(ADP-ribose) polymerase/PARP1 and PARP2 identified using a cell-based screen in yeast

Cancer Research

Volumn 61, Issue 10, 2001, Pages 4175-4183

  Perkins, E ^a   Sun, D ^a   Nguyen, A ^a   Tulac, S ^a   Francesco, M ^a   Tavana, H ^a   Nguyen, H ^a   Tugendreich, S ^a   Barthmaier, P ^a   Couto, J ^a   Yeh, E ^a   Thode, S ^a   Jarnagin, K ^a   Jain, A ^a   Morgans, D ^a   Melese, T ^a  

^a Entelos Inc   (United States)

Author keywords

[No Author keywords available]

Indexed keywords

6(5H) PHENANTHRIDINONE; GLYCOSIDASE; NICOTINAMIDE ADENINE DINUCLEOTIDE ADENOSINE DIPHOSPHATE RIBOSYLTRANSFERASE; PHENANTHRIDINE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; ENZYME ACTIVE SITE; ENZYME INHIBITION; GENE MUTATION; HUMAN; NONHUMAN; PRIORITY JOURNAL; PROTEIN EXPRESSION; PROTEIN FAMILY; SACCHAROMYCES CEREVISIAE; VALIDATION PROCESS;

ATP-BINDING CASSETTE TRANSPORTERS; BINDING SITES; DRUG EVALUATION, PRECLINICAL; ENZYME INHIBITORS; GENE EXPRESSION; HUMANS; ISOENZYMES; MEMBRANE PROTEINS; MUTATION; PHENANTHRENES; POLY(ADP-RIBOSE) POLYMERASES; SACCHAROMYCES CEREVISIAE; SACCHAROMYCES CEREVISIAE PROTEINS;

EID: 0035872473     PISSN: 00085472     EISSN: None     Source Type: Journal    
DOI: None     Document Type: Article

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