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Volumn 428, Issue 2, 2001, Pages 177-184
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Efficacy of antipsychotic agents at human 5-HT1A receptors determined by [3H]WAY100,635 binding affinity ratios: Relationship to efficacy for G-protein activation
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Author keywords
5 HT1A receptor; Antipsychotic; Clozapine; Inverse agonist; S16924; WAY100,635
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Indexed keywords
1 [2 [4 (6 FLUORO 1,2 BENZISOXAZOL 3 YL) 1 PIPERIDYL]ETHYL] 3 PHENYL 2 IMIDAZOLINONE;
ALPHA (4 FLUOROPHENYL) 4 (5 FLUORO 2 PYRIMIDINYL) 1 PIPERAZINEBUTANOL;
ALPHA [1 [2 (1,4 BENZODIOXAN 5 YLOXY)ETHYL] 3 PYRROLIDINYL] 4 FLUOROACETOPHENONE;
BUTACLAMOL;
CHLORPROMAZINE;
CLOZAPINE;
GUANINE NUCLEOTIDE BINDING PROTEIN;
GUANOSINE 5' O (3 THIOTRIPHOSPHATE);
HALOPERIDOL;
LIGAND;
LOXAPINE;
N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE;
NEUROLEPTIC AGENT;
OCAPERIDONE;
OLANZAPINE;
QUETIAPINE;
RISPERIDONE;
SEROTONIN 1A RECEPTOR;
SPIPERONE;
SULFUR 35;
THIORIDAZINE;
TIOSPIRONE;
TRITIUM;
UNCLASSIFIED DRUG;
ZIPRASIDONE;
ANIMAL CELL;
ARTICLE;
BINDING AFFINITY;
CHO CELL;
CONTROLLED STUDY;
DRUG ACTIVITY;
DRUG DETERMINATION;
DRUG EFFICACY;
DRUG RECEPTOR BINDING;
DRUG SELECTIVITY;
NONHUMAN;
PRIORITY JOURNAL;
RECEPTOR OCCUPANCY;
ANIMALS;
ANTIPSYCHOTIC AGENTS;
BINDING, COMPETITIVE;
CHLORPROMAZINE;
CHO CELLS;
CLOZAPINE;
CRICETINAE;
DOSE-RESPONSE RELATIONSHIP, DRUG;
GTP-BINDING PROTEINS;
GUANOSINE 5'-O-(3-THIOTRIPHOSPHATE);
HALOPERIDOL;
HUMANS;
MEMBRANES;
PIPERAZINES;
PIPERIDINES;
PYRIDINES;
PYRIMIDINONES;
PYRROLIDINES;
RECEPTORS, SEROTONIN;
RECEPTORS, SEROTONIN, 5-HT1;
THIAZOLES;
THIORIDAZINE;
TRITIUM;
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EID: 0035812644
PISSN: 00142999
EISSN: None
Source Type: Journal
DOI: 10.1016/S0014-2999(01)01344-9 Document Type: Article |
Times cited : (23)
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References (43)
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