Thiazole and thiadiazole analogues as a novel class of adenosine receptor antagonists

Journal of Medicinal Chemistry

Volumn 44, Issue 5, 2001, Pages 749-762

  Van Muijlwijk Koezen, J E ^a   Timmerman, H ^a   Vollinga, R C ^b   Frijtag von Drabbe Kunzel J ^b   De Groote, M ^b   Visser, S ^a   IJzerman, A P ^b  

^a VU UNIVERSITY AMSTERDAM   (Netherlands)

^b LEIDEN UNIVERSITY   (Netherlands)

Author keywords

[No Author keywords available]

Indexed keywords

4 HYDROXYBENZAMIDE; ADENOSINE; ADENOSINE RECEPTOR BLOCKING AGENT; HETEROCYCLIC COMPOUND; THIADIAZOLE DERIVATIVE; THIAZOLE DERIVATIVE; UNCLASSIFIED DRUG;

ARTICLE; BINDING AFFINITY; CIS TRANS ISOMERISM; MOLECULAR RECOGNITION; PROTEIN ANALYSIS; STEREOCHEMISTRY; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS;

ANIMALS; BRAIN; CYCLOHEXYLAMINES; MODELS, MOLECULAR; MOLECULAR CONFORMATION; RADIOLIGAND ASSAY; RATS; RECEPTOR, ADENOSINE A2A; RECEPTOR, ADENOSINE A3; RECEPTORS, PURINERGIC P1; STRUCTURE-ACTIVITY RELATIONSHIP; THIADIAZOLES; THIAZOLES;

EID: 0035282632     PISSN: 00222623     EISSN: None     Source Type: Journal    
DOI: 10.1021/jm0003945     Document Type: Article

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