SCOPUS 정보 검색 플랫폼

Volumn 9, Issue 7, 2001, Pages 1753-1764

Molecular modeling, structure-activity relationships and functional antagonism studies of 4-hydroxy-1-methyl-4-(4-methylphenyl)-3-piperidyl 4-methylphenyl ketones as a novel class of dopamine transporter inhibitors

(6) Wang, Shaomeng a Sakamuri, Sukumar a Enyedy, Istvan J a Kozikowski, Alan P a Zaman, Wahiduz A b Johnson, Kenneth M b

a GEORGETOWN UNIVERSITY MEDICAL CENTER (United States)

b University of Texas Medical Branch School of Medicine (United States)

Author keywords

[No Author keywords available]

Indexed keywords

4 HYDROXY 1 METHYL 4 (4 METHYLPHENYL) 3 PIPERIDYL 4 METHYLPHENYLKETONE; 4 HYDROXY 1 METHYL 4 (4 METHYLPHENYL) 3 PIPERIDYL 4 METHYLPHENYLKETONE DERIVATIVE; COCAINE; DOPAMINE TRANSPORTER; DOPAMINE UPTAKE INHIBITOR; MAZINDOL; NORADRENALIN TRANSPORTER; SEROTONIN TRANSPORTER; TRITIUM; UNCLASSIFIED DRUG;

AMINE TRANSPORT; ANIMAL TISSUE; ARTICLE; BRAIN CORTEX; CARBON NUCLEAR MAGNETIC RESONANCE; CHIRALITY; CONTROLLED STUDY; CORPUS STRIATUM; DOPAMINE UPTAKE; DRUG ANTAGONISM; DRUG SELECTIVITY; DRUG SYNTHESIS; ENANTIOMER; HIGH PERFORMANCE LIQUID CHROMATOGRAPHY; ISOMER; MOLECULAR MODEL; NONHUMAN; PROTON NUCLEAR MAGNETIC RESONANCE; RACEMIC MIXTURE; RAT; SEROTONIN UPTAKE; STRUCTURE ACTIVITY RELATION;

ANIMALS; CARRIER PROTEINS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; CORPUS STRIATUM; DOPAMINE; DOPAMINE PLASMA MEMBRANE TRANSPORT PROTEINS; MAGNETIC RESONANCE SPECTROSCOPY; MEMBRANE GLYCOPROTEINS; MEMBRANE TRANSPORT PROTEINS; MODELS, MOLECULAR; NERVE TISSUE PROTEINS; NOREPINEPHRINE; PIPERIDINES; RATS; SEROTONIN; STRUCTURE-ACTIVITY RELATIONSHIP; SYNAPTOSOMES;

EID: 0034944353 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00090-6 Document Type: Article

Times cited : (19)

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