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Volumn 64, Issue 7, 2001, Pages 874-882

The complestatins as HIV-1 integrase inhibitors. Efficient isolation, structure elucidation, and inhibitory activities of isocomplestatin, chloropeptin I, new complestatins, A and B, and acid-hydrolysis products of chloropeptin I

(13) Singh, S B a Jayasuriya, H a Salituro, G M a Zink, D L a Shafiee, A a Heimbuch, B a Silverman, K C a Lingham, R B a Genilloud, O b Teran, A b Vilella, D b Felock, P a Hazuda, D a

a MERCK RESEARCH LABORATORIES (United States)

b Medical affairs Merck sharp and Dohme ltd (Spain)

Author keywords

[No Author keywords available]

Indexed keywords

CHLOROPEPTIN I; COMPLESTATIN; COMPLESTATIN A; COMPLESTATIN B; INTEGRASE; INTEGRASE INHIBITOR; ISOCOMPLESTATIN; UNCLASSIFIED DRUG;

ARTICLE; CHIRALITY; DRUG ACTIVITY; DRUG ISOLATION; DRUG STRUCTURE; ENZYME ACTIVITY; ENZYME INHIBITION; HUMAN IMMUNODEFICIENCY VIRUS 1; HYDROLYSIS; IC 50; ISOMER; NONHUMAN; PH; REVERSED PHASE LIQUID CHROMATOGRAPHY; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS; VIRUS REPLICATION;

ANTI-HIV AGENTS; ANTIGENS, CD45; CHLOROPHENOLS; CHROMATOGRAPHY, HIGH PRESSURE LIQUID; GAS CHROMATOGRAPHY-MASS SPECTROMETRY; HIV ENVELOPE PROTEIN GP120; HIV INTEGRASE; HIV INTEGRASE INHIBITORS; HIV-1; MAGNETIC RESONANCE SPECTROSCOPY; MODELS, CHEMICAL; MOLECULAR STRUCTURE; OLIGOPEPTIDES; PEPTIDES, CYCLIC; STEREOISOMERISM; STREPTOMYCES; STRUCTURE-ACTIVITY RELATIONSHIP;

HUMAN IMMUNODEFICIENCY VIRUS; HUMAN IMMUNODEFICIENCY VIRUS 1;

EID: 0034899584 PISSN: 01633864 EISSN: None Source Type: Journal
DOI: 10.1021/np000632z Document Type: Article

Times cited : (94)

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