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Volumn 9, Issue 10, 2001, Pages 2683-2691

Synthesis and evaluation of diazine containing bioisosteres of (-)-ferruginine as ligands for nicotinic acetylcholine receptors

(6) Gundisch D a Harms, K a Schwarz, S a Seitz, G a Stubbs, M T a Wegge, T a

a PHILIPPS UNIVERSITY MARBURG (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

2 (4 PYRIDAZINYL) 8 AZABICYCLO[3.2.1]OCT 2 ENE; 2 (5 PYRIMIDINYL) 8 AZABICYCLO[3.2.1]OCT 2 ENE; 2 (TRIFLUOROMETHANESULFONYLOXY) 8 AZABICYCLO[3.2.1]OCT 2 ENE 8 CARBOXYLIC ACID ETHYL ESTER; 2 TROPANONE; ACETIC ACID DERIVATIVE; ANATOXIN A; EPIBATIDINE; FERRUGININE; LIGAND; NICOTINE; NICOTINIC RECEPTOR; PYRAZINE; PYRIDAZINE; PYRIMIDINE; RECEPTOR SUBTYPE; SULFADIAZINE; TRIBUTYLSTANNYL DIAZEPINE; UNCLASSIFIED DRUG; VINYLTRIFLATE;

BINDING AFFINITY; CATALYSIS; CATALYST; CHEMICAL REACTION; CHIRALITY; CONFERENCE PAPER; DIAGNOSTIC TEST; DRUG SELECTIVITY; DRUG SYNTHESIS; ENANTIOMER; EVALUATION; REACTION ANALYSIS; SPECTROSCOPY; STRUCTURE ACTIVITY RELATION; STRUCTURE ANALYSIS; X RAY CRYSTALLOGRAPHY;

ANIMALS; BACTERIAL TOXINS; BICYCLO COMPOUNDS, HETEROCYCLIC; BRAIN; CATALYSIS; CHROMATOGRAPHY, THIN LAYER; CRYSTALLOGRAPHY, X-RAY; LIGANDS; MARINE TOXINS; MESYLATES; MICROCYSTINS; MOLECULAR CONFORMATION; MOLECULAR STRUCTURE; NICOTINE; ORGANOTIN COMPOUNDS; PALLADIUM; PYRIDINES; RATS; RATS, SPRAGUE-DAWLEY; RECEPTORS, NICOTINIC; SPECTROPHOTOMETRY, ULTRAVIOLET; STEREOISOMERISM; STRUCTURE-ACTIVITY RELATIONSHIP; TROPANES; VINYL COMPOUNDS;

EID: 0034842156 PISSN: 09680896 EISSN: None Source Type: Journal
DOI: 10.1016/S0968-0896(01)00188-2 Document Type: Article

Times cited : (26)

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