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1
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0029914328
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For a recent review, see
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For a recent review, see: Mansell, H. L. Tetrahedron 1996, 52, 6025-6061.
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Mansell, H.L.1
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3
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0034614434
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-
For the most recent syntheses, see: (a)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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(2000)
Tetrahedron
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, pp. 309-315
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Parsons, P.J.1
Camp, N.P.2
Edwards, N.3
Sumoreeah, L.R.4
-
4
-
-
0342278581
-
-
(b)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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(1999)
Angew. Chem.
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, pp. 2178-2180
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-
Aggarwal, V.L.1
Humphries, P.S.2
Fenwick, A.3
-
5
-
-
0033549543
-
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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Angew. Chem., Int. Ed. Engl.
, vol.38
, pp. 1985-1986
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-
-
6
-
-
0033531676
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-
(c)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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(1999)
J. Am. Chem. Soc.
, vol.121
, pp. 3057-3064
-
-
Trost, B.M.1
Oslob, J.D.2
-
7
-
-
0032499133
-
-
(d)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
-
(1998)
Tetrahedron Lett.
, vol.39
, pp. 2133-2136
-
-
Oh, C.-Y.1
Kim, K.-S.2
Ham, W.-A.3
-
8
-
-
33748649334
-
-
(e)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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(1997)
J. Chem. Soc., Perkin Trans.
, vol.1
, pp. 2313-2318
-
-
Magnus, N.A.1
Ducry, L.2
Rolland, V.3
Wonnacott, S.4
Gallagher, T.5
-
9
-
-
0030603125
-
-
(f)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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(1996)
Tetrahedron
, vol.52
, pp. 11637-11642
-
-
Parsons, P.J.1
Camp, N.P.2
Underwood, J.M.3
Harvey, D.M.4
-
10
-
-
0029026296
-
-
(g)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
-
(1995)
J. Chem. Soc., Chem. Commun.
, pp. 831-832
-
-
Newcombe, N.J.1
Simpkins, N.S.2
-
11
-
-
0001260134
-
-
(h)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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J. Org. Chem.
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-
-
Hernandez, A.1
Rapoport, H.2
-
12
-
-
0001204816
-
-
(i)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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J. Org. Chem.
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Sardine, F.J.1
Howard, M.H.2
Morningstar, M.3
Rapoport, H.4
-
13
-
-
0022214795
-
-
(j)
-
For the most recent syntheses, see: (a) Parsons, P. J.; Camp, N. P.; Edwards, N.; Sumoreeah, L. R. Tetrahedron 2000, 56, 309-315; (b) Aggarwal, V. L.; Humphries, P. S.; Fenwick. A. Angew. Chem. 1999, 111, 2178-2180; Angew. Chem., Int. Ed. Engl. 1999, 38, 1985-1986; (c) Trost, B. M.; Oslob, J. D. J. Am. Chem. Soc. 1999, 121, 3057-3064; (d) Oh, C.-Y.; Kim, K.-S.; Ham, W.-A.; Tetrahedron Lett. 1998, 39, 2133-2136; (e) Magnus, N. A.; Ducry, L.; Rolland, V.; Wonnacott, S.; Gallagher, T. J. Chem. Soc., Perkin Trans. 1 1997, 2313-2318; (f) Parsons, P. J.; Camp. N. P.; Underwood, J. M.; Harvey, D. M. Tetrahedron 1996, 52, 11637-11642; (g) Newcombe, N. J.; Simpkins, N. S. J. Chem. Soc., Chem. Commun. 1995, 831-832; (h) Hernandez, A.; Rapoport, H. J. Org. Chem. 1994, 59, 1058-1066; (i) Sardine, F. J.; Howard, M. H.; Morningstar, M.; Rapoport, H. J. Org. Chem. 1990, 55, 5025-5033; (j) Koskinen, A. M. P.; Rapoport, H. J. Med. Chem. 1985, 28, 1301-1309.
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Koskinen, A.M.P.1
Rapoport, H.2
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14
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0031450275
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For recent reviews on nAChRs as targets for drug discovery, see: (a)
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For recent reviews on nAChRs as targets for drug discovery, see: (a) Holladay, M. W.; Dart, M. J.; Lynch, J. K. J. Med. Chem. 1998, 40, 4169-4194; (b) Holladay, M. W.; Lebold, S. A.; Lin, N.-H. Drug Dev. Res. 1995, 35, 191-213.
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Lynch, J.K.3
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15
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0029119941
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(b)
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For recent reviews on nAChRs as targets for drug discovery, see: (a) Holladay, M. W.; Dart, M. J.; Lynch, J. K. J. Med. Chem. 1998, 40, 4169-4194; (b) Holladay, M. W.; Lebold, S. A.; Lin, N.-H. Drug Dev. Res. 1995, 35, 191-213.
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For leading references, see: (a) Podlech, J.; J. Prakt. Chem. 1998, 340, 679-682; (b) Yang, S.; Hungerhoff, B.; Metz, P.; Tetrahedron Lett. 1998, 39, 2097-2098.
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Podlech, J.1
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0032499095
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(b)
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For leading references, see: (a) Podlech, J.; J. Prakt. Chem. 1998, 340, 679-682; (b) Yang, S.; Hungerhoff, B.; Metz, P.; Tetrahedron Lett. 1998, 39, 2097-2098.
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Tetrahedron Lett.
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Yang, S.1
Hungerhoff, B.2
Metz, P.3
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