Antagonistic action of a 25-carboxylic ester analogue of 1α,25- dihydroxyvitamin D3 is mediated by a lack of ligand-induced vitamin D receptor interaction with coactivators

Journal of Biological Chemistry

Volumn 275, Issue 22, 2000, Pages 16506-16512

  Herdick, Michaela ^a   Steinmeyer, Andreas ^b   Carlberg, Carsten ^a  

^a HEINRICH HEINE UNIVERSITY   (Germany)

^b BAYER PHARMA AG   (Germany)

Author keywords

[No Author keywords available]

Indexed keywords

1,3,24 TRIHYDROXY 26,27 CYCLO 9,10 SECOCHOLESTA 5,7,10(19),22 TETRAENE 25 CARBOXYLIC ACID BUTYL ESTER; BUTYL 1,3,24 TRIHYDROXY 26,27 CYCLO 9,10 SECOCHOLESTA 5,7,10(19),22 TETRAENE 25 CARBOXYLIC ACID; CALCITRIOL; CALCITRIOL DERIVATIVE; RETINOID X RECEPTOR; UNCLASSIFIED DRUG; VITAMIN D RECEPTOR;

ARTICLE; COMPETITIVE INHIBITION; CONTROLLED STUDY; DRUG ANTAGONISM; DRUG RECEPTOR BINDING; DRUG STRUCTURE; IN VITRO STUDY; IN VIVO STUDY; PRIORITY JOURNAL; PROTEIN PROTEIN INTERACTION;

EID: 0034595679     PISSN: 00219258     EISSN: None     Source Type: Journal    
DOI: 10.1074/jbc.M910000199     Document Type: Article

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