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Nuclear Medicine and Biology

Volumn 27, Issue 5, 2000, Pages 441-447

A retrospect on the discovery of WAY-100635 and the prospect for improved 5-HT(1A) receptor PET radioligands

(1) Cliffe, Ian A a

a Vernalis PLC (United Kingdom)

Author keywords

5 HT(1A) Receptors; Carbon 11; CPC 222; FEC; FPC; NAD 299; p MPPF; PET; WAY 100635

Indexed keywords

CPC 222; FLUOROBENZENE; N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDYL)CYCLOHEXANECARBOXAMIDE; NOR N [2 [4 (2 METHOXYPHENYL) 1 PIPERAZINYL]ETHYL] N (2 PYRIDINYL) 2 BICYCLO[2 2 2] OCTANE CARBOXAMIDE; RADIOLIGAND; ROBALZOTAN; SEROTONIN 1A ANTAGONIST; SEROTONIN 1A RECEPTOR; TRANS FLUOROCYCLOHEXANE; UNCLASSIFIED DRUG;

BRAIN TOMOGRAPHY; CHEMICAL ANALYSIS; CHEMICAL MODIFICATION; CHEMICAL STRUCTURE; HUMAN; ISOTOPE LABELING; LIGAND BINDING; POSITRON EMISSION TOMOGRAPHY; REVIEW; STOICHIOMETRY; STRUCTURE ACTIVITY RELATION;

EID: 0033831097 PISSN: 09698051 EISSN: None Source Type: Journal
DOI: 10.1016/S0969-8051(00)00109-8 Document Type: Article

Times cited : (42)

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