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Bioorganic and Medicinal Chemistry Letters

Volumn 10, Issue 18, 2000, Pages 2119-2122

Design, synthesis, and discovery of 3-piperazinyl-3,4-dihydro-2(1H)-quinolinone derivatives: A novel series of mixed dopamine D2/D4 receptor antagonists

(5) Zhao, He a Thurkauf, Andrew a Braun, Julia a Brodbeck, Robin a Kieltyka, Andrzej a

a NEUROGEN CORPORATION (United States)

Author keywords

[No Author keywords available]

Indexed keywords

CLOZAPINE; DOPAMINE 2 RECEPTOR; DOPAMINE 2 RECEPTOR BLOCKING AGENT; DOPAMINE 4 RECEPTOR; EMONAPRIDE; GAMMA LACTAM DERIVATIVE; LACTAM; PRAZOSIN; QUINOLONE DERIVATIVE;

ANIMAL TISSUE; ARTICLE; DRUG DESIGN; DRUG RECEPTOR BINDING; DRUG SYNTHESIS; NONHUMAN; RAT; STRUCTURE ACTIVITY RELATION;

ANTIPSYCHOTIC AGENTS; CLOZAPINE; HUMANS; LACTAMS; PIPERAZINES; PROTEIN BINDING; QUINOLONES; RECEPTORS, DOPAMINE; RECEPTORS, DOPAMINE D2; RECEPTORS, DOPAMINE D4; STRUCTURE-ACTIVITY RELATIONSHIP;

ANIMALIA;

EID: 0033813482 PISSN: 0960894X EISSN: None Source Type: Journal
DOI: 10.1016/S0960-894X(00)00421-2 Document Type: Article

Times cited : (40)

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