Pharmacology of cloned human 5-HT1D receptor-mediated functional responses in stably transfected rat C6-glial cell lines: Further evidence differentiating human 5-HT1D and 5-HT1B receptors

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 353, Issue 2, 1996, Pages 144-156

  Pauwels, Petrus J ^a   Palmier, Christiane ^a   Wurch, Thierry ^a   Colpaert, Francis C ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

Agonist antagonist; cAMP; Cell growth; Cloned human 5 HT1D 5 HT1B receptor; Permanent transfection; Rat C6 glial cell line

Indexed keywords

1 (3 TRIFLUOROMETHYLPHENYL)PIPERAZINE; 1 NAPHTHYLPIPERAZINE; 2 DIPROPYLAMINO 8 HYDROXYTETRALIN; 4 (4 METHYL 1 PIPERAZINYL) 7 TRIFLUOROMETHYLPYRROLO[1,2 A]QUINOXALINE; 5 CARBAMOYLTRYPTAMINE; 5 METHOXY 3 (1,2,3,6 TETRAHYDRO 4 PYRIDYL) 1H INDOLE; 5 METHOXYTRYPTAMINE; BUFOTENINE; COMPLEMENTARY DNA; CYCLIC AMP; FORSKOLIN; KETANSERIN; MESSENGER RNA; METERGOLINE; METITEPINE; N [4 METHOXY 3 (4 METHYL 1 PIPERAZINYL)PHENYL] 2' METHYL 4' (5 METHYL 1,2,4 OXADIAZOL 3 YL)[1,1' BIPHENYL] 4 CARBOXAMIDE; PARTIAL AGONIST; RADIOLIGAND; RITANSERIN; SEROTONIN; SEROTONIN 1B RECEPTOR; SEROTONIN 1D RECEPTOR; SEROTONIN AGONIST; SEROTONIN ANTAGONIST; SUMATRIPTAN; TRYPTAMINE; UNCLASSIFIED DRUG;

ANIMAL CELL; ARTICLE; BINDING AFFINITY; CELL GROWTH; CELL LINE; CONTROLLED STUDY; DRUG POTENCY; GENETIC TRANSFECTION; GLIA CELL; HUMAN; LIGAND BINDING; MOLECULAR CLONING; NONHUMAN; PLASMID; RAT; RECEPTOR DENSITY; RECEPTOR INTRINSIC ACTIVITY; REVERSE TRANSCRIPTION POLYMERASE CHAIN REACTION;

ANIMALS; BINDING, COMPETITIVE; CELL LINE; DOSE-RESPONSE RELATIONSHIP, DRUG; HUMANS; KETANSERIN; NEUROGLIA; RATS; RECEPTORS, SEROTONIN; RITANSERIN; RNA, MESSENGER;

EID: 0030052084     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/BF00168751     Document Type: Article

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