Interaction of 5-HT(1B/D) ligands recombinant h 5-HT(1A) receptors: Intrinsic activity and modulation by G-protein activation state

Naunyn-Schmiedeberg's Archives of Pharmacology

Volumn 357, Issue 5, 1998, Pages 490-499

  Pauwels, Petrus J ^a   Palmier, Christiane ^a   Dupuis, Delphine S ^a   Colpaert, Francis C ^a  

^a INSTITUT DE RECHERCHE PIERRE FABRE   (France)

Author keywords

5 HT(1B D) agonists; 35S GTP S binding response; C6 glial and HeLa cell lines; Ligand efficacy; Recombinant h 5 HT(1A) receptor

Indexed keywords

2 DIPROPYLAMINO 8 HYDROXYTETRALIN; CP 122638; DIHYDROERGOTAMINE; FLESINOXAN; GUANINE NUCLEOTIDE BINDING PROTEIN; NARATRIPTAN; RIZATRIPTAN; SEROTONIN 1A RECEPTOR; SUMATRIPTAN; UNCLASSIFIED DRUG; ZOLMITRIPTAN; GUANOSINE DIPHOSPHATE; LISURIDE; RECOMBINANT PROTEIN; SEROTONIN AGONIST; SEROTONIN RECEPTOR;

ARTICLE; CELL MEMBRANE; CONTROLLED STUDY; HELA CELL; HUMAN; HUMAN CELL; LIGAND BINDING; RECEPTOR BINDING; RECEPTOR DENSITY; DRUG EFFECT; GLIA; METABOLISM; RADIOASSAY;

CELL MEMBRANE; DIHYDROERGOTAMINE; GTP-BINDING PROTEINS; GUANOSINE DIPHOSPHATE; HELA CELLS; HUMANS; LISURIDE; NEUROGLIA; RADIOLIGAND ASSAY; RECEPTORS, SEROTONIN; RECOMBINANT PROTEINS; SEROTONIN AGONISTS;

EID: 0031595667     PISSN: 00281298     EISSN: None     Source Type: Journal    
DOI: 10.1007/PL00005198     Document Type: Article

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