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See, for example: (a) Gordeev, M. F.; Patel, D. V.; Gordon, E. M. J. Org. Chem. 1996, 61, 924. (b) Mjalli, A. M. M.; Sarshar, S.; Baiga, T. J. Tetrahedron Lett. 1996, 37, 2943. (c) Hutchins, S. M.; Chapman, K. T. Tetrahedron Lett. 1996, 37, 4869. (d) Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643. (e) Kolodziej, S. A.; Hamper, B. C. Tetrahedron Lett. 1996, 37, 5277. (f) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937.
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Mjalli, A.M.M.1
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See, for example: (a) Gordeev, M. F.; Patel, D. V.; Gordon, E. M. J. Org. Chem. 1996, 61, 924. (b) Mjalli, A. M. M.; Sarshar, S.; Baiga, T. J. Tetrahedron Lett. 1996, 37, 2943. (c) Hutchins, S. M.; Chapman, K. T. Tetrahedron Lett. 1996, 37, 4869. (d) Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643. (e) Kolodziej, S. A.; Hamper, B. C. Tetrahedron Lett. 1996, 37, 5277. (f) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937.
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See, for example: (a) Gordeev, M. F.; Patel, D. V.; Gordon, E. M. J. Org. Chem. 1996, 61, 924. (b) Mjalli, A. M. M.; Sarshar, S.; Baiga, T. J. Tetrahedron Lett. 1996, 37, 2943. (c) Hutchins, S. M.; Chapman, K. T. Tetrahedron Lett. 1996, 37, 4869. (d) Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643. (e) Kolodziej, S. A.; Hamper, B. C. Tetrahedron Lett. 1996, 37, 5277. (f) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937.
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See, for example: (a) Gordeev, M. F.; Patel, D. V.; Gordon, E. M. J. Org. Chem. 1996, 61, 924. (b) Mjalli, A. M. M.; Sarshar, S.; Baiga, T. J. Tetrahedron Lett. 1996, 37, 2943. (c) Hutchins, S. M.; Chapman, K. T. Tetrahedron Lett. 1996, 37, 4869. (d) Gordeev, M. F.; Patel, D. V.; Wu, J.; Gordon, E. M. Tetrahedron Lett. 1996, 37, 4643. (e) Kolodziej, S. A.; Hamper, B. C. Tetrahedron Lett. 1996, 37, 5277. (f) Dressman, B. A.; Spangle, L. A.; Kaldor, S. W. Tetrahedron Lett. 1996, 37, 937.
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44
-
-
85033147792
-
-
note
-
14 (bp 56°C; price $389/1 gal).
-
-
-
-
46
-
-
85033151615
-
-
note
-
1H NMR spectrum of orthothioester 4 we could always observe some fluorous impurities. Attempts to purify 4 were not successful.
-
-
-
-
47
-
-
85033133235
-
-
note
-
Reactions were usually run on 0.5-0.7 mmol scale. If the reaction sequence was performed on a larger scale, a decrease in the yield was observed.
-
-
-
-
48
-
-
85033140513
-
-
For Ugi reactions on solid polymer supports, see ref 17
-
For Ugi reactions on solid polymer supports, see ref 17.
-
-
-
-
49
-
-
85033149427
-
-
NMR spectra of acid 7 were recorded in neat deuterated trifluoroacetic acid
-
NMR spectra of acid 7 were recorded in neat deuterated trifluoroacetic acid.
-
-
-
-
51
-
-
0642316448
-
-
New Orleans, 1996; American Chemical Society: Washington, DC, ORGN 122
-
For a related solid-phase modification of the Biginelli reaction, see: Robinett, L. D.; Yager, K. M.; Phelan, J. C. 211th National Meeting of the American Chemical Society, New Orleans, 1996; American Chemical Society: Washington, DC, 1996; ORGN 122.
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(1996)
211th National Meeting of the American Chemical Society
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-
Robinett, L.D.1
Yager, K.M.2
Phelan, J.C.3
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