New antiestrogens from a library screen of homoallylic amides, allylic amides, and C-cyclopropylalkylamides

Bioorganic and Medicinal Chemistry

Volumn 13, Issue 1, 2005, Pages 157-164

  Janjic, Jelena M ^a   Mu, Ying ^a   Kendall, Christopher ^a   Stephenson, Corey R J ^a   Balachandran, Raghavan ^a   Raccor, Brianne S ^a   Lu, Ying ^a   Zhu, Guangyu ^a   Xie, Wen ^a   Wipf, Peter ^a   Day, Billy W ^a  

^a UNIVERSITY OF PITTSBURGH   (United States)

Author keywords

Cell based screen; Estrogen receptor ; Estrogen response element; Fluorescent estrogen; Transcription

Indexed keywords

AMIDE; ANTIESTROGEN; CARBAMIC ACID DERIVATIVE; TAMOXIFEN;

ARTICLE; BREAST CANCER; CANCER CELL CULTURE; CELL PROLIFERATION; CELL STRAIN MCF 7; CONTROLLED STUDY; CYTOTOXICITY; DRUG ACTIVITY; DRUG IDENTIFICATION; DRUG SCREENING; ENANTIOMER; HUMAN; HUMAN CELL;

AMIDES; CELL LINE; CELL LINE, TUMOR; DRUG SCREENING ASSAYS, ANTITUMOR; ESTROGEN RECEPTOR MODULATORS; GENES, REPORTER; HUMANS; RECEPTORS, ESTROGEN; STRUCTURE-ACTIVITY RELATIONSHIP;

MINK CELL FOCUS-FORMING VIRUS; STAPHYLOCOCCUS PHAGE 3A;

EID: 9644303168     PISSN: 09680896     EISSN: None     Source Type: Journal    
DOI: 10.1016/j.bmc.2004.09.048     Document Type: Article

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