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Angewandte Chemie - International Edition

Volumn 55, Issue 40, 2016, Pages 12479-12483

Partially Saturated Bicyclic Heteroaromatics as an sp3-Enriched Fragment Collection

(7) Twigg, David G a Kondo, Noriyasu a,b Mitchell, Sophie L a Galloway, Warren R J D a Sore, Hannah F a Madin, Andrew c Spring, David R a

a UNIVERSITY OF CAMBRIDGE (United Kingdom)

b SHIONOGI AND CO LTD (Japan)

c ASTRAZENECA (United Kingdom)

Author keywords

drug design; drug discovery; fused ring systems; nitrogen heterocycles; synthetic methods

Indexed keywords

SCAFFOLDS;

DRUG DESIGN; DRUG DISCOVERY; FUSED-RING SYSTEM; NITROGEN HETEROCYCLES; SYNTHETIC METHODS;

LEAD COMPOUNDS;

EID: 84985994996 PISSN: 14337851 EISSN: 15213773 Source Type: Journal
DOI: 10.1002/anie.201606496 Document Type: Article

Times cited : (52)

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